SCHEMBL7414012

SCHEMBL7414012

O=C(O)CCn1c(=O)ncc2ccc(O)cc21

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMO O15229 6/20 0.43
WEE1 P30291 2/20 0.41
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
HTR2B P41595 1/20 0.40
ALDH1A1 P00352 1/20 0.39
FABP3 P05413 1/20 0.39
FABP4 P15090 1/20 0.39
FABP5 Q01469 1/20 0.39
APEX1 P27695 1/20 0.38
MAPT P10636 1/20 0.38
CHEK1 O14757 1/20 0.38
SRC P12931 1/20 0.38
KDM4E B2RXH2 2/20 0.37
LMNA P02545 1/20 0.37
KMT2A Q03164 1/20 0.37
POLB P06746 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7415741 0.89 WEE1 (0.44) KMOWEE1ALDH1A1FABP3FABP4
SCHEMBL10621833 0.81 KMO (0.57) KMOALDH1A1FABP3FABP4FABP5
Iodide SCHEMBL10619045 0.80 KMO (0.56) KMOALDH1A1FABP3FABP4FABP5
SCHEMBL10747226 0.76 TBXAS1 (0.42) KMOALDH1A1FABP3FABP4FABP5
SCHEMBL7405683 0.76 KMO (0.45) KMOWEE1ALDH1A1FABP3FABP4
SCHEMBL7412024 0.73 WEE1 (0.50) KMOWEE1ALDH1A1FABP3FABP4
SCHEMBL7418131 0.73 KMO (0.41) KMOWEE1ALDH1A1FABP3FABP4
SCHEMBL7405656 0.72 FABP4 (0.45) WEE1ALDH1A1FABP3FABP4FABP5
SCHEMBL7414631 0.70 DYRK1A (0.54) KMO
SCHEMBL7407798 0.70 WEE1 (0.47) KMOWEE1ALDH1A1FABP3FABP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4631283-A RENAL VASODILATORS, CARDIOVASCULAR AGENTS ORTHO PHARMACEUTICAL CORPORATION (US) 1986-12-23 US disclosed
US-4490374-A CARDIOVASCULAR AGENTS ORTHO PHARMACEUTICAL CORPORATION (US) 1984-12-25 US disclosed
EP-0107398-A1 Ortho substituted dihydroxy-2(1H)quinazolinone-1-alkanoic acids ORTHO PHARMACEUTICAL CORPORATION (US) 1984-05-02 EP disclosed