SCHEMBL7415741

SCHEMBL7415741

O=C(O)CCn1c(=O)ncc2cc(O)ccc21

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
WEE1 P30291 4/20 0.44
KMO O15229 5/20 0.43
ALDH1A1 P00352 1/20 0.42
CHEK1 O14757 2/20 0.40
SRC P12931 1/20 0.40
KDM4E B2RXH2 3/20 0.39
POLB P06746 1/20 0.39
HSD17B10 Q99714 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
FABP3 P05413 1/20 0.39
FABP4 P15090 1/20 0.39
FABP5 Q01469 1/20 0.39
APEX1 P27695 2/20 0.38
MAPT P10636 1/20 0.38
LMNA P02545 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7414012 0.89 KMO (0.43) WEE1KMOALDH1A1CHEK1SRC
SCHEMBL10747226 0.82 TBXAS1 (0.42) KMOALDH1A1SRCKDM4EPOLB
SCHEMBL10621833 0.81 KMO (0.57) KMOALDH1A1KDM4EPOLBL3MBTL1
Iodide SCHEMBL10619045 0.80 KMO (0.56) KMOALDH1A1KDM4EPOLBL3MBTL1
SCHEMBL7412024 0.76 WEE1 (0.50) WEE1KMOALDH1A1CHEK1SRC
SCHEMBL7405656 0.75 FABP4 (0.45) WEE1ALDH1A1CHEK1SRCKDM4E
SCHEMBL7405683 0.73 KMO (0.45) WEE1KMOALDH1A1CHEK1SRC
SCHEMBL7407798 0.73 WEE1 (0.47) WEE1KMOALDH1A1CHEK1SRC
SCHEMBL7405772 0.70 DYRK1A (0.51) KMOALDH1A1KDM4EHSD17B10L3MBTL1
SCHEMBL7418131 0.70 KMO (0.41) WEE1KMOALDH1A1CHEK1SRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4631283-A RENAL VASODILATORS, CARDIOVASCULAR AGENTS ORTHO PHARMACEUTICAL CORPORATION (US) 1986-12-23 US disclosed
US-4490374-A CARDIOVASCULAR AGENTS ORTHO PHARMACEUTICAL CORPORATION (US) 1984-12-25 US disclosed
EP-0107398-A1 Ortho substituted dihydroxy-2(1H)quinazolinone-1-alkanoic acids ORTHO PHARMACEUTICAL CORPORATION (US) 1984-05-02 EP disclosed