SCHEMBL7414191

SCHEMBL7414191

Cc1cc(C)c(C)c(S(=O)(=O)Nc2cccc3c2N(C(=O)CCc2ccc(C#N)cc2)CCC3)c1C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.42
TP53 P04637 1/20 0.39
ALDH1A1 P00352 5/20 0.38
MEN1 O00255 3/20 0.38
HPGD P15428 3/20 0.38
KMT2A Q03164 3/20 0.38
KDM4E B2RXH2 2/20 0.38
HSD17B10 Q99714 2/20 0.38
CRHBP P24387 1/20 0.38
CRHR2 Q13324 1/20 0.38
MAPT P10636 3/20 0.36
NPSR1 Q6W5P4 1/20 0.36
NR3C1 P04150 1/20 0.36
GLA P06280 1/20 0.35
GAA P10253 1/20 0.35
POLB P06746 2/20 0.35
HDAC1 Q13547 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
USP2 O75604 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6983600 0.92 MAPT (0.40) PKMTP53ALDH1A1MEN1KMT2A
SCHEMBL7411038 0.87 PKM (0.43) PKMTP53ALDH1A1MEN1KMT2A
SCHEMBL6985749 0.87 ALDH1A1 (0.48) PKMTP53ALDH1A1MEN1KMT2A
SCHEMBL6985322 0.85 GAA (0.41) PKMTP53ALDH1A1MEN1KMT2A
SCHEMBL6978509 0.84 PTGER4 (0.40) ALDH1A1MEN1HPGDKMT2AHSD17B10
SCHEMBL6977498 0.84 CCKBR (0.44) PKMTP53ALDH1A1MEN1KMT2A
SCHEMBL6984039 0.84 TP53 (0.45) PKMTP53ALDH1A1KDM4EMAPT
SCHEMBL6984851 0.83 BRD4 (0.50) PKMTP53MEN1KMT2AMAPT
SCHEMBL7408050 0.83 TP53 (0.40) PKMTP53ALDH1A1MEN1HPGD
SCHEMBL6982764 0.83 FPR1 (0.43) PKMALDH1A1MEN1HPGDKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT Boehringer Ingelheim Pharma KG (DE) 2000-04-12 EP disclosed
WO-1999000371-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-01-07 WO disclosed