SCHEMBL6982764

SCHEMBL6982764

N#Cc1ccc(CCC(=O)N2CCCc3cccc(NS(=O)(=O)c4ccc(F)cc4)c32)cc1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
FPR1 P21462 3/20 0.43
FPR2 P25090 3/20 0.43
GAA P10253 3/20 0.40
METAP2 P50579 1/20 0.39
PKM P14618 2/20 0.39
SLC16A3 O15427 1/20 0.39
ALDH1A1 P00352 6/20 0.39
SMN1; SMN2 Q16637 3/20 0.39
LMNA P02545 1/20 0.39
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
SLC22A12 Q96S37 1/20 0.38
KDM4E B2RXH2 1/20 0.38
HPGD P15428 1/20 0.38
HSD17B10 Q99714 1/20 0.38
MAPT P10636 2/20 0.38
MCOLN3 Q8TDD5 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
NR3C1 P04150 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6985322 0.92 GAA (0.41) FPR1FPR2GAAMETAP2PKM
SCHEMBL7408050 0.92 TP53 (0.40) GAAPKMALDH1A1SMN1; SMN2LMNA
SCHEMBL6985749 0.92 ALDH1A1 (0.48) GAAPKMALDH1A1LMNAMEN1
SCHEMBL6984759 0.92 LMNA (0.47) GAAPKMALDH1A1SMN1; SMN2LMNA
SCHEMBL6981764 0.90 METAP2 (0.42) GAAMETAP2PKMSLC16A3ALDH1A1
SCHEMBL6981583 0.89 STAT3 (0.49) GAAPKMSLC16A3ALDH1A1SMN1; SMN2
SCHEMBL6982163 0.88 SLC16A3 (0.45) GAAPKMSLC16A3ALDH1A1SMN1; SMN2
SCHEMBL6977498 0.87 CCKBR (0.44) GAAPKMALDH1A1LMNAMEN1
SCHEMBL7411038 0.87 PKM (0.43) GAAPKMALDH1A1SMN1; SMN2LMNA
SCHEMBL6984039 0.87 TP53 (0.45) GAAPKMALDH1A1LMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed
EP-0991624-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT Boehringer Ingelheim Pharma KG (DE) 2000-04-12 EP disclosed
WO-1999000371-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-01-07 WO disclosed