SCHEMBL7424092

SCHEMBL7424092

CC(C)C[C@@H](C(=O)O)N(CCc1ccc(-c2cccnc2)cc1)C(=O)O

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PSMB5 P28074 3/20 0.49
MKNK1 Q9BUB5 3/20 0.44
MKNK2 Q9HBH9 3/20 0.44
GPR88 Q9GZN0 1/20 0.43
NTSR1 P30989 1/20 0.42
PRCP P42785 1/20 0.41
MMP12 P39900 2/20 0.41
CYP2A6 P11509 1/20 0.41
CTSL P07711 1/20 0.41
CTSS P25774 1/20 0.41
CTSK P43235 1/20 0.41
ADAMTS4 O75173 1/20 0.41
WNT3A P56704 1/20 0.40
AKR1C3 P42330 1/20 0.40
AKR1C2 P52895 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7425766 1.00 PSMB5 (0.49) PSMB5MKNK1MKNK2GPR88NTSR1
SCHEMBL7427409 0.88 MMP12 (0.46) GPR88MMP12CTSLCTSSCTSK
SCHEMBL7420384 0.88 MMP12 (0.46) GPR88MMP12CTSLCTSSCTSK
SCHEMBL7421351 0.82 MMP13 (0.48) PSMB5ADAMTS4
SCHEMBL7424796 0.82 HPGD (0.38) GPR88
SCHEMBL7425601 0.81 MCHR1 (0.50) GPR88
SCHEMBL7378945 0.80 MEN1 (0.48)
SCHEMBL7424495 0.80 HCAR2 (0.43) GPR88CTSLCTSK
SCHEMBL7419478 0.78 MMP2 (0.42) AKR1C2
SCHEMBL7424015 0.78 GPR88 (0.42) GPR88CTSLCTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002039997-A2 ACE-2 MODULATING COMPOUNDS AND USE THEREOF MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-05-23 WO disclosed