SCHEMBL742529

SCHEMBL742529

COCCCn1c(C2(O)CCCN(C(=O)OC(C)(C)C)C2)nc2ccccc21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 2/20 0.40
CCR5 P51681 3/20 0.39
TSHR P16473 1/20 0.38
PIN1 Q13526 1/20 0.38
CYP11B2 P19099 1/20 0.37
ADORA2A P29274 2/20 0.37
OPRM1 P35372 1/20 0.37
OPRD1 P41143 1/20 0.37
OGFRL1 Q5TC84 1/20 0.37
HPGD P15428 2/20 0.37
MMP3 P08254 1/20 0.37
MMP7 P09237 1/20 0.37
MMP10 P09238 1/20 0.37
MMP8 P22894 1/20 0.37
MMP12 P39900 1/20 0.37
REN P00797 2/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
GLA P06280 1/20 0.36
GAA P10253 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL738785 0.81 GPR119 (0.35) CYP11B2
SCHEMBL741974 0.78 KCNH2 (0.52)
SCHEMBL741975 0.78 KCNH2 (0.52)
SCHEMBL7954887 0.77 KDM4E (0.47) CCR5TSHRKDM4EALDH1A1HSD17B10
SCHEMBL742271 0.75 REN (0.44) TSHROPRM1OPRD1HPGDREN
SCHEMBL7627768 0.72 ALDH1A1 (0.55) OPRM1OPRD1OGFRL1ALDH1A1
SCHEMBL6982730 0.71 TSHR (0.47) TSHRCYP11B2OPRD1
SCHEMBL31513766 0.71 TSHR (0.47) TSHRCYP11B2OPRD1
SCHEMBL7629372 0.70 ALDH1A1 (0.52) ALDH1A1
SCHEMBL21359237 0.69 SIGMAR1 (0.44) TSHRCYP11B2OPRM1OPRD1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed
US-8138168-B1 Renin inhibitors TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2012-03-20 US disclosed