SCHEMBL7426883

SCHEMBL7426883

COc1cccc(S(=O)(=O)N2CCCC(NC(=O)CCC(C)C)C(=O)C2)c1

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PAX8 Q06710 1/20 0.43
CTSK P43235 2/20 0.42
ALDH1A1 P00352 3/20 0.42
LMNA P02545 2/20 0.42
NPSR1 Q6W5P4 2/20 0.42
TP53 P04637 1/20 0.42
HTT P42858 1/20 0.42
MAPT P10636 2/20 0.42
HCRTR1 O43613 1/20 0.42
HCRTR2 O43614 1/20 0.42
CHRM5 P08912 1/20 0.42
PKM P14618 3/20 0.41
GAA P10253 2/20 0.41
PKLR P30613 1/20 0.41
POLB P06746 1/20 0.41
CTSL P07711 1/20 0.40
CTSS P25774 1/20 0.40
MTNR1A P48039 1/20 0.40
MTNR1B P49286 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7431356 0.88 KMT2A (0.46) CTSKALDH1A1LMNAHTTMAPT
SCHEMBL7599077 0.85 HCRTR1 (0.40) CTSKALDH1A1LMNANPSR1TP53
SCHEMBL7426881 0.85 HDAC1 (0.42) PAX8CTSKALDH1A1LMNANPSR1
SCHEMBL7427486 0.82 MEN1 (0.47) CTSKALDH1A1LMNAGAAPOLB
SCHEMBL7434831 0.82 KMT2A (0.48) ALDH1A1NPSR1TP53MAPTPKM
SCHEMBL7432035 0.79 ALDH1A1 (0.48) CTSKALDH1A1CTSLCTSS
Quinoxaline SCHEMBL5099608 0.79 CTSK (0.49) CTSKCHRM5PKMCTSLCTSS
SCHEMBL7477927 0.79 CTSK (0.50) CTSKLMNAMAPTCTSLCTSS
SCHEMBL4772275 0.78 MTNR1A (0.40) ALDH1A1MTNR1AMTNR1B
SCHEMBL7427121 0.78 MEN1 (0.55) ALDH1A1HTTMAPTHCRTR1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1158986-A4 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2002-03-27 EP claimed
EP-1158986-A1 PROTEASE INHIBITORS SmithKline Beecham Corporation (US) 2001-12-05 EP claimed
WO-2000038687-A1 PROTEASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2000-07-06 WO claimed