SCHEMBL7427147

SCHEMBL7427147

CC(C)C[C@@H](C(=O)N(C)CC#N)N(C(=O)c1ccccc1)c1csc(N2CCNCC2)n1

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CTSL P07711 14/20 0.46
CTSS P25774 14/20 0.46
CTSB P07858 13/20 0.46
CTSK P43235 12/20 0.46
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
BAZ2A Q9UIF9 1/20 0.35
CHEK1 O14757 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7488490 0.83 CTSK (0.48) CTSLCTSSCTSBCTSK
SCHEMBL7427146 0.74 CTSL (0.49) CTSLCTSSCTSBCTSKNPC1
SCHEMBL6184317 0.73 CTSS (0.56) CTSLCTSSCTSBCTSK
SCHEMBL6184312 0.70 CTSL (0.54) CTSLCTSSCTSBCTSKNPC1
SCHEMBL7451296 0.67 CTSL (0.47) CTSLCTSSCTSBCTSK
SCHEMBL7486127 0.65 CTSK (0.55) CTSLCTSSCTSBCTSKNPC1
SCHEMBL7439201 0.64 CTSK (0.62) CTSLCTSSCTSBCTSKNPC1
SCHEMBL7650560 0.64 CTSB (0.49) CTSLCTSSCTSBCTSKNPC1
SCHEMBL6185770 0.64 CTSK (0.56) CTSLCTSSCTSBCTSK
SCHEMBL4714257 0.63 CTSL (1.00) CTSLCTSSCTSBCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001068645-A2 N-CYANOMETHYLCARBOXAMIDES AND THEIR USE AS PROTEASE INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2001-09-20 WO claimed