SCHEMBL7433904

SCHEMBL7433904

COc1ccc(CC(CC(O)C(N)CC2CCCCC2)C(=O)O)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LDHA P00338 1/20 0.45
METAP2 P50579 3/20 0.45
METAP1 P53582 2/20 0.45
CPB2 Q96IY4 1/20 0.44
EPHX2 P34913 2/20 0.41
PPARG P37231 2/20 0.41
DPP4 P27487 1/20 0.41
FAP Q12884 1/20 0.41
DPP8 Q6V1X1 1/20 0.41
DPP9 Q86TI2 1/20 0.41
DPP7 Q9UHL4 1/20 0.41
REN P00797 3/20 0.40
KMT2A Q03164 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
HPGD P15428 1/20 0.40
CYP2C19 P33261 1/20 0.40
MMP1 P03956 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7433911 1.00 LDHA (0.45) LDHAMETAP2METAP1CPB2EPHX2
Hydrochloric Acid SCHEMBL9876367 0.88 MMP1 (0.47) METAP2METAP1CPB2EPHX2REN
SCHEMBL8894601 0.86 MME (0.43) METAP2METAP1PPARGRENANPEP
SCHEMBL8894607 0.86 MME (0.43) METAP2METAP1PPARGRENANPEP
SCHEMBL7430623 0.85 METAP2 (0.45) METAP2METAP1PPARGDPP4FAP
SCHEMBL7430616 0.85 METAP2 (0.45) METAP2METAP1PPARGDPP4FAP
SCHEMBL8891774 0.84 LDHA (0.56) LDHAPPARGKMT2ACYP1A2CYP2D6
SCHEMBL8891766 0.84 LDHA (0.56) LDHAPPARGKMT2ACYP1A2CYP2D6
SCHEMBL7436178 0.83 EPHX1 (0.42) METAP2METAP1PPARGDPP4FAP
SCHEMBL7444348 0.83 DPEP1 (0.44) METAP2METAP1EPHX2PPARGDPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5643878-A TREATMENT OF RETROVIRAL DISEASES LIKE AIDS CIBA-GEIGY CORPORATION (US) 1997-07-01 US disclosed
EP-0618222-A2 Dipeptid derivatives of 5-amino-4-hydroxy-hexanoic acid CIBA-GEIGY AG (CH) 1994-10-05 EP disclosed
EP-0532466-A2 Derivatives of 5-amino-4-hydroxy-hexanoic acid and their therapeutical use CIBA-GEIGY AG (CH) 1993-03-17 EP disclosed