SCHEMBL7434681

SCHEMBL7434681

CSc1ccc2c(c1)OCC(C=O)O2

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
ALDH1A1 P00352 6/20 0.35
SMN1; SMN2 Q16637 3/20 0.35
LMNA P02545 3/20 0.35
NPC1 O15118 2/20 0.33
MAPT P10636 2/20 0.33
RAB9A P51151 2/20 0.33
TP53 P04637 2/20 0.33
TSHR P16473 2/20 0.33
POLB P06746 1/20 0.33
NFKB1 P19838 1/20 0.33
NFKB2 Q00653 1/20 0.33
RELA Q04206 1/20 0.33
PDE5A O76074 2/20 0.31
ITGB2 P05107 2/20 0.31
ICAM1 P05362 2/20 0.31
ITGAL P20701 2/20 0.31
KDM4E B2RXH2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7434823 0.80 AR (0.37) ALDH1A1SMN1; SMN2LMNANPC1RAB9A
SCHEMBL7437340 0.80 CA2 (0.42) KMT2ANPC1RAB9AMAOB
SCHEMBL7443159 0.76 CA2 (0.48) HCRTR2NPC1MAOB
SCHEMBL2487394 0.76 CA2 (0.48) HCRTR2NPC1MAOB
SCHEMBL7434686 0.76 NPC1 (0.42) HCRTR2MEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL7445863 0.76 MTNR1A (0.44) MEN1KMT2AALDH1A1SMN1; SMN2LMNA
SCHEMBL7437879 0.75 DAO (0.41) HCRTR2ALDH1A1NPC1MAPTRAB9A
SCHEMBL7436261 0.74 ALDH1A1 (0.32) ALDH1A1SMN1; SMN2NPC1MAPTRAB9A
SCHEMBL1299583 0.73 NISCH (0.44) ALDH1A1SMN1; SMN2NPC1RAB9APOLB
SCHEMBL1299611 0.73 NISCH (0.44) ALDH1A1SMN1; SMN2NPC1RAB9APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4558129-A Benzodioxanyl-hydroxyethylene-piperazinyl acetanilides which effect calcium entry and β-blockade SYNTEX (U.S.A.) INC. (US) 1985-12-10 US disclosed
US-4499100-A CARDIOUVASCULAR DISORDERS SYNTEX (U.S.A.) INC. (US) 1985-02-12 US disclosed