SCHEMBL7436642

SCHEMBL7436642

CC(C)CC(CNC(Cc1ccccc1)C(=O)CSCc1ccco1)NC(=O)CCC1CCCCC1

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.42
HPGD P15428 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
BCHE P06276 1/20 0.41
POLB P06746 1/20 0.39
PSMB5 P28074 4/20 0.38
PSMB1 P20618 1/20 0.38
PSMB2 P49721 1/20 0.38
REN P00797 6/20 0.37
MMP3 P08254 2/20 0.37
MMP1 P03956 1/20 0.37
MMP2 P08253 1/20 0.37
EPHX2 P34913 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7444403 0.95 BCHE (0.42) ALDH1A1HPGDSMN1; SMN2BCHEPOLB
SCHEMBL7313879 0.88 ALDH1A1 (0.44) ALDH1A1HPGDSMN1; SMN2PSMB5PSMB1
SCHEMBL7436647 0.88 ALDH1A1 (0.44) ALDH1A1HPGDSMN1; SMN2PSMB5PSMB1
SCHEMBL7301739 0.88 ALDH1A1 (0.43) ALDH1A1HPGDSMN1; SMN2POLBPSMB5
SCHEMBL7437241 0.87 ALDH1A1 (0.39) ALDH1A1HPGDSMN1; SMN2BCHEPOLB
SCHEMBL7312132 0.86 CTSG (0.43) ALDH1A1HPGDSMN1; SMN2POLBPSMB5
SCHEMBL8680990 0.85 ALDH1A1 (0.40) ALDH1A1HPGDSMN1; SMN2POLBPSMB5
SCHEMBL7299047 0.84 PSEN1 (0.44) ALDH1A1HPGDSMN1; SMN2BCHEPSMB5
SCHEMBL7444412 0.84 PSEN1 (0.44) ALDH1A1HPGDSMN1; SMN2BCHEPSMB5
SCHEMBL7303357 0.82 CTSS (0.46) ALDH1A1POLBPSMB5PSMB1PSMB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0525420-B1 Pseudopeptides and dipeptides characterised by a substituted methyl ketone moiety at the C-terminus as thiol protease inhibitors MITSUBISHI CHEM CORP (JP) 1999-05-12 EP disclosed
US-5834508-A PROTEASE ENZYME INHIBITORS; MUSCLE DISORDERS MITSUBISHI CHEMICAL CORPORATION (JP) 1998-11-10 US disclosed
US-5639783-A POTENT PROTEASE INHIBITOR FOR TREATING MUSCULAR, NERVOUS SYSTEM DISEASES MITSUBISHI CHEMICAL CORPORATION (JP) 1997-06-17 US disclosed