SCHEMBL7441165

SCHEMBL7441165

NC(=O)c1nc(-c2cc(Cl)cc(Cl)c2)cs1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
SCN9A Q15858 1/20 0.44
RAB9A P51151 3/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
ATP4A P20648 2/20 0.41
ATP4B P51164 2/20 0.41
CDC7 O00311 1/20 0.41
DBF4 Q9UBU7 1/20 0.41
ALOX5 P09917 1/20 0.41
MAP3K14 Q99558 1/20 0.40
ABL1 P00519 2/20 0.40
KMO O15229 1/20 0.38
ENPP2 Q13822 2/20 0.38
ROCK1 Q13464 1/20 0.38
GSTO1 P78417 1/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
ALDH1A1 P00352 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6664214 0.84 ATP4A (0.60) CYP3A4CYP2D6CYP2C9SCN9ARAB9A
SCHEMBL2734989 0.83 RAB9A (0.54) CYP3A4RAB9ASMN1; SMN2ALOX5ABL1
SCHEMBL7429957 0.81 ATP4A (0.43) RAB9ASMN1; SMN2ATP4AATP4BALOX5
SCHEMBL7440680 0.80 ABL1 (0.57) RAB9AALOX5ABL1MEN1KMT2A
SCHEMBL16238595 0.76 CYP3A4 (0.50) CYP3A4CYP2D6CYP2C9SCN9ARAB9A
SCHEMBL168593 0.76 ALDH1A1 (0.56) CYP3A4CYP2D6CYP2C9SCN9ARAB9A
SCHEMBL3088513 0.76 MAP2K3 (0.50) CYP3A4CYP2D6CYP2C9SCN9ARAB9A
SCHEMBL5999257 0.75 KDM4E (0.55) RAB9ASMN1; SMN2CDC7DBF4MEN1
SCHEMBL7436623 0.75 PKM (0.55) CYP3A4CYP2D6CYP2C9SCN9ARAB9A
SCHEMBL7438064 0.75 MAPT (0.43) CYP3A4CYP2D6CYP2C9SCN9AMAP3K14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0506194-B1 4-aryl-thiazole or imidazole derivatives AKZO NOBEL NV (NL) 1996-08-21 EP disclosed
US-5462959-A 4-aryl-imidazole derivatives AKZO N.V. (NL) 1995-10-31 US disclosed
US-5254575-A 4-aryl-thiazole derivatives AKZO N.V. (NL) 1993-10-19 US disclosed
EP-0506194-A1 4-aryl-thiazole or imidazole derivatives Akzo Nobel N.V. (NL) 1992-09-30 EP disclosed