SCHEMBL7445894

SCHEMBL7445894

CC(C)c1ccc(N)c(-c2ccc(F)c(Cl)c2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 6/20 0.42
PTGS1 P23219 4/20 0.42
SLC1A3 P43003 1/20 0.41
SLC1A2 P43004 1/20 0.41
SLC1A1 P43005 1/20 0.41
EPHB4 P54760 2/20 0.41
PGR P06401 1/20 0.40
APP P05067 2/20 0.40
PSEN1 P49768 1/20 0.40
PSEN2 P49810 1/20 0.40
APH1B Q8WW43 1/20 0.40
NCSTN Q92542 1/20 0.40
APH1A Q96BI3 1/20 0.40
PSENEN Q9NZ42 1/20 0.40
ALDH1A1 P00352 2/20 0.39
CYP3A4 P08684 1/20 0.39
TSHR P16473 1/20 0.39
MAPK1 P28482 1/20 0.39
GAA P10253 1/20 0.39
ALOX12 P18054 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7444699 0.85 AHR (0.46) PTGS1APPPSEN1PSEN2APH1B
SCHEMBL7442456 0.83 ADRB2 (0.44) PTGS1ALDH1A1CYP3A4TSHRMAPK1
SCHEMBL7446405 0.81 PTGS2 (0.44) PTGS2PTGS1SLC1A3SLC1A2SLC1A1
SCHEMBL3388331 0.80 PTGS2 (0.46) PTGS2PTGS1EPHB4ALDH1A1CYP3A4
SCHEMBL530400 0.79 SLC6A2 (0.44) PTGS2PTGS1PGRALDH1A1CYP3A4
SCHEMBL17486766 0.79 SLC6A2 (0.44) PTGS2PTGS1PGRALDH1A1CYP3A4
SCHEMBL14041057 0.76 RXRA (0.49) PTGS2PTGS1PGRCYP3A4TSHR
SCHEMBL29901014 0.75 ALDH1A1 (0.56) PTGS1ALDH1A1GAAALOX12HTT
SCHEMBL31161110 0.75 PTGS2 (0.58) PTGS2PTGS1EPHB4ALDH1A1CYP3A4
SCHEMBL12618445 0.75 LMNA (0.42) PTGS2PTGS1APPPSEN1PSEN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0691966-B1 QUINOLINES AS TYPE IV PHOSPHODIESTERASE INHIBITORS SYNTEX INC (US) 1998-09-09 EP disclosed
WO-1994022852-A1 QUINOLINES AS TYPE IV PHOSPHODIESTERASE INHIBITORS SYNTEX (U.S.A.) INC. (US) 1994-10-13 WO disclosed