SCHEMBL7448981

SCHEMBL7448981

Cc1c(S(=O)(=O)N2CCCC2)ccc2[nH]c(COc3cccc(C#N)c3)nc12

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.43
HTR2C P28335 2/20 0.43
HPGD P15428 1/20 0.38
HTT P42858 3/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
MCOLN3 Q8TDD5 1/20 0.38
FFAR1 O14842 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
GAA P10253 2/20 0.36
MAPT P10636 2/20 0.36
LMNA P02545 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
POLB P06746 1/20 0.36
MMP13 P45452 1/20 0.36
MMP14 P50281 1/20 0.36
FABP1 P07148 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7396002 0.76 CKS1B (0.49) ALDH1A1HTTMEN1KMT2ATDP1
SCHEMBL7394535 0.74 CKS1B (0.49) ALDH1A1HTTMEN1KMT2AGAA
SCHEMBL7419866 0.72 RAB9A (0.44) ALDH1A1HTR2CHTTMEN1KMT2A
SCHEMBL6782097 0.69 HTR2C (0.50) ALDH1A1HTR2CHTTLMNASMN1; SMN2
SCHEMBL7379409 0.67 SMN1; SMN2 (0.42) ALDH1A1HTTMEN1KMT2AFFAR1
SCHEMBL7445307 0.67 TGFBR1 (0.40) ALDH1A1HPGDMAPTLMNASMN1; SMN2
SCHEMBL7393202 0.65 SMN1; SMN2 (0.42) ALDH1A1HTTMEN1KMT2ATDP1
SCHEMBL23882572 0.64 ROCK2 (0.61) ALDH1A1HTTMEN1KMT2AGAA
SCHEMBL30947514 0.63 PDE9A (0.56)
SCHEMBL15550259 0.63 PDE9A (0.56)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0966454-A1 DISUBSTITUTED BICYCLIC HETEROCYCLES, THEIR PRODUCTION AND USE AS MEDICAMENTS Boehringer Ingelheim Pharma KG (DE) 1999-12-29 EP disclosed
WO-1998037075-A1 DISUBSTITUTED BICYCLIC HETEROCYCLES, THEIR PRODUCTION AND USE AS MEDICAMENTS BOEHRINGER INGELHEIM PHARMA KG (DE) 1998-08-27 WO disclosed