SCHEMBL7453286

SCHEMBL7453286

COc1ccc(S(=O)(=O)N(C)CC(=O)N[C@@H](Cc2ccc3ccccc3c2)C(=O)O)cc1OC

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4D Q08499 2/20 0.55
ALDH1A1 P00352 6/20 0.52
MAPK1 P28482 1/20 0.52
KMT2A Q03164 2/20 0.52
CA2 P00918 1/20 0.51
HCRTR1 O43613 1/20 0.50
HCRTR2 O43614 1/20 0.50
FPR2 P25090 1/20 0.48
TP53 P04637 1/20 0.48
PIN1 Q13526 1/20 0.47
L3MBTL1 Q9Y468 2/20 0.47
MAPT P10636 2/20 0.47
HTT P42858 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
MEN1 O00255 1/20 0.47
HSD17B10 Q99714 1/20 0.47
MME P08473 1/20 0.46
ACE P12821 1/20 0.46
CPA1 P15085 1/20 0.46
ACE2 Q9BYF1 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7514233 0.84 MME (0.49) PDE4DALDH1A1CA2HCRTR1HCRTR2
SCHEMBL7447456 0.82 MME (0.56) PDE4DCA2HCRTR1HCRTR2FPR2
SCHEMBL7444546 0.78 MMP13 (0.52) ALDH1A1KMT2ACA2FPR2PIN1
SCHEMBL7916012 0.76 MME (0.58) KMT2ACA2FPR2MEN1MME
SCHEMBL5572753 0.75 SMN1; SMN2 (0.55) ALDH1A1MAPK1KMT2AHTTSMN1; SMN2
SCHEMBL6375346 0.74 ITGA4 (0.46) ALDH1A1KMT2ACA2FPR2HTT
SCHEMBL757454 0.73 MME (0.62) CA2PIN1MMEACECPA1
SCHEMBL2779203 0.73 MME (0.62) CA2PIN1MMEACECPA1
SCHEMBL28067038 0.73 LDHA (0.64) ALDH1A1MAPK1KMT2AFPR2MAPT
SCHEMBL10663094 0.72 FPR2 (0.61) ALDH1A1MAPK1KMT2AFPR2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6221888-B1 ANTIHISTAMINE, ANTIINFLAMMATORY AGENT, AUTOIMMUNE DISEASE, RHEUMATIC DISORDERS MERCK & CO., INC. 2001-04-24 US claimed
EP-0998282-A4 SULFONAMIDES AS CELL ADHESION INHIBITORS MERCK & CO INC (US) 2000-08-30 EP claimed
EP-0998282-A1 SULFONAMIDES AS CELL ADHESION INHIBITORS Merck & Co., Inc. (a New Jersey corp.) (US) 2000-05-10 EP claimed
WO-1998053818-A1 SULFONAMIDES AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1998-12-03 WO claimed