SCHEMBL7447456

SCHEMBL7447456

CC[C@H](C)[C@@H](C(=O)N[C@@H](Cc1ccc2ccccc2c1)C(=O)O)N(C)S(=O)(=O)c1ccc(OC)c(OC)c1

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MME P08473 13/20 0.56
ACE P12821 11/20 0.56
CPA1 P15085 9/20 0.56
ACE2 Q9BYF1 9/20 0.56
CA2 P00918 1/20 0.46
PDE4D Q08499 1/20 0.45
FPR2 P25090 1/20 0.44
PIN1 Q13526 1/20 0.42
ITGB3 P05106 1/20 0.42
ITGAV P06756 1/20 0.42
MMP1 P03956 1/20 0.42
MMP9 P14780 1/20 0.42
MMP13 P45452 1/20 0.42
ADAM17 P78536 1/20 0.42
HCRTR1 O43613 1/20 0.42
HCRTR2 O43614 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7514233 0.93 MME (0.49) MMEACECPA1ACE2CA2
SCHEMBL7916012 0.83 MME (0.58) MMEACECPA1ACE2CA2
SCHEMBL7453286 0.82 PDE4D (0.55) MMEACECPA1ACE2CA2
SCHEMBL7444546 0.79 MMP13 (0.52) MMEACECPA1ACE2CA2
SCHEMBL7447863 0.77 MME (0.51) MMEACECPA1ACE2CA2
SCHEMBL7447944 0.77 MME (0.52) MMEACECPA1ACE2CA2
SCHEMBL7452231 0.75 MME (0.50) MMEACECPA1ACE2CA2
SCHEMBL7446281 0.72 FPR2 (0.45) MMEACECPA1ACE2PDE4D
SCHEMBL7447599 0.71 CA2 (0.44) MMECA2PDE4DITGB3ITGAV
SCHEMBL6375346 0.69 ITGA4 (0.46) CA2FPR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6221888-B1 ANTIHISTAMINE, ANTIINFLAMMATORY AGENT, AUTOIMMUNE DISEASE, RHEUMATIC DISORDERS MERCK & CO., INC. 2001-04-24 US claimed
EP-0998282-A4 SULFONAMIDES AS CELL ADHESION INHIBITORS MERCK & CO INC (US) 2000-08-30 EP claimed
EP-0998282-A1 SULFONAMIDES AS CELL ADHESION INHIBITORS Merck & Co., Inc. (a New Jersey corp.) (US) 2000-05-10 EP claimed
WO-1998053818-A1 SULFONAMIDES AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1998-12-03 WO claimed