SCHEMBL7458396

SCHEMBL7458396

NCc1ccc(N2CC(C(=O)[C@@H](Cc3ccccc3)C(=O)O)OC2=O)cc1

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 9/20 0.43
MAOA P21397 1/20 0.37
ANPEP P15144 1/20 0.36
ERAP1 Q9NZ08 1/20 0.36
PTPN1 P18031 1/20 0.36
ADORA2A P29274 1/20 0.36
ALDH1A1 P00352 1/20 0.34
PKM P14618 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7461978 0.81 MAOA (0.44) GRM2MAOA
SCHEMBL8892282 0.80 NAMPT (0.41) ADORA2A
SCHEMBL7465489 0.74 MEN1 (0.42) ALDH1A1
SCHEMBL8891141 0.72 ITGB3 (0.40) GRM2ALDH1A1
SCHEMBL28023734 0.72 FADS1 (0.60) GRM2
SCHEMBL7461829 0.71 ITGB3 (0.45) MAOA
SCHEMBL5762328 0.71 GRM2 (0.53) GRM2MAOA
SCHEMBL7457894 0.70 MAOA (0.36) GRM2MAOA
SCHEMBL7462123 0.70 ADORA2A (0.48) ADORA2A
SCHEMBL8893573 0.70 ADORA2A (0.48) GRM2PTPN1ADORA2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0697408-B1 1 substituted-phenyl-oxazolidene-2-one derivatives and their use as adhesion-receptor antagonists MERCK PATENT GMBH (DE) 2002-01-23 EP disclosed
US-5614535-A Adhesion receptor antagonists MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1997-03-25 US disclosed
EP-0697408-A1 1 substituted-phenyl-oxazolidene-2-one derivatives and their use as adhesion-receptor antagonists MERCK PATENT GmbH (DE) 1996-02-21 EP disclosed