SCHEMBL7464929

SCHEMBL7464929

O=C(Cc1ccncc1)N1CCC(c2c[nH]c3ccc(F)cc23)CC1

nearest known ligand 0.57

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 5/20 0.57
OPRM1 P35372 2/20 0.52
OPRK1 P41145 2/20 0.52
OPRL1 P41146 2/20 0.52
NMT2 O60551 1/20 0.51
NMT1 P30419 1/20 0.51
GRM5 P41594 1/20 0.51
CCR2 P41597 3/20 0.49
SLC6A4 P31645 3/20 0.48
HTR1A P08908 2/20 0.48
HTR1D P28221 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8556742 0.85 HSD11B1 (0.61) HSD11B1OPRM1OPRK1OPRL1CCR2
SCHEMBL5340537 0.80 HSD11B1 (0.68) HSD11B1OPRM1OPRK1OPRL1CCR2
Hydrochloric Acid SCHEMBL9049559 0.79 OPRM1 (0.59) OPRM1OPRK1OPRL1SLC6A4HTR1A
SCHEMBL18324763 0.79 KDM4E (0.69) HSD11B1OPRM1OPRK1OPRL1SLC6A4
SCHEMBL27510903 0.77 HSD11B1 (0.51) HSD11B1OPRM1OPRK1OPRL1CCR2
SCHEMBL6347867 0.76 HSD11B1 (0.76) HSD11B1OPRM1OPRK1OPRL1CCR2
SCHEMBL10922885 0.75 HSD11B1 (0.66) HSD11B1OPRM1OPRK1OPRL1CCR2
SCHEMBL18324845 0.75 DRD2 (0.61) HSD11B1OPRM1OPRK1OPRL1CCR2
SCHEMBL8557474 0.75 HSD11B1 (0.48) HSD11B1OPRM1OPRK1OPRL1CCR2
SCHEMBL22605559 0.74 ALDH1A1 (0.58) HSD11B1CCR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0708102-B1 5-HT1F agonists for the treatment of migraine LILLY CO ELI (US) 2002-12-11 EP disclosed
US-5721252-A PIPERIDINYL-1H-INDOLE DERIVATIVES ELI LILLY AND COMPANY (US) 1998-02-24 US disclosed
US-5521196-A ANALGESICS USING SEROTONIN ANTAGONIST ELI LILLY AND COMPANY (US) 1996-05-28 US disclosed
EP-0708102-A1 5-HT1F agonists for the treatment of migraine ELI LILLY AND COMPANY (US) 1996-04-24 EP disclosed