SCHEMBL7467427

SCHEMBL7467427

O=c1c2ccc(Cl)cc2n(Cc2ccccn2)c(=O)n1S(=O)(=O)c1ccc(Cl)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.47
AGTR1 P30556 1/20 0.47
PARG Q86W56 2/20 0.44
CMA1 P23946 1/20 0.43
GABRA1 P14867 3/20 0.43
GABRA5 P31644 3/20 0.43
MEN1 O00255 1/20 0.42
GAA P10253 1/20 0.42
KMT2A Q03164 1/20 0.42
LMNA P02545 1/20 0.41
NOX4 Q9NPH5 3/20 0.41
GRIN1 Q05586 1/20 0.40
GRIN2B Q13224 1/20 0.40
MAPK8 P45983 1/20 0.39
MAPK9 P45984 1/20 0.39
PSEN1 P49768 1/20 0.39
PSEN2 P49810 1/20 0.39
APH1B Q8WW43 1/20 0.39
NCSTN Q92542 1/20 0.39
APH1A Q96BI3 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7460713 0.85 MAPK8 (0.55) ALDH1A1CMA1MEN1GAAKMT2A
SCHEMBL7466124 0.83 CMA1 (0.46) PARGCMA1GABRA1GABRA5GRIN1
SCHEMBL7463810 0.81 SMN1; SMN2 (0.45) ALDH1A1MEN1KMT2ALMNAPSEN1
SCHEMBL4456863 0.80 GABRA5 (0.53) PARGCMA1GABRA1GABRA5KMT2A
SCHEMBL7469901 0.80 CMA1 (0.44) ALDH1A1PARGCMA1GAALMNA
SCHEMBL7461329 0.78 CMA1 (0.46) ALDH1A1PARGCMA1MEN1KMT2A
SCHEMBL7463851 0.78 NOX4 (0.46) ALDH1A1PARGCMA1MEN1GAA
SCHEMBL7459226 0.76 PARG (0.44) ALDH1A1PARGCMA1MEN1KMT2A
SCHEMBL7468517 0.76 HDAC6 (0.52) CMA1MEN1KMT2AMAPK8MAPK9
SCHEMBL7462052 0.76 KMT2A (0.47) ALDH1A1PARGCMA1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0795548-B1 QUINAZOLINE DERIVATIVES AND USE THEREOF SUNTORY LTD (JP) 2002-07-03 EP disclosed
US-5814631-A CHYMASE INHIBITOR, CARDIVASCULAR SUNTORY LIMITED (JP) 1998-09-29 US disclosed
EP-0795548-A1 QUINAZOLINE DERIVATIVES AND USE THEREOF SUNTORY LIMITED (JP) 1997-09-17 EP disclosed