SCHEMBL7459226

SCHEMBL7459226

N#Cc1ccc(Cn2c(=O)n(S(=O)(=O)c3ccc(Cl)cc3)c(=O)c3ccc(Cl)cc32)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARG Q86W56 4/20 0.44
CMA1 P23946 1/20 0.44
HDAC6 Q9UBN7 4/20 0.42
HDAC1 Q13547 3/20 0.42
HDAC8 Q9BY41 3/20 0.42
SRC P12931 2/20 0.41
MAPK8 P45983 1/20 0.40
MAPK9 P45984 1/20 0.40
P2RX3 P56373 1/20 0.39
PRKACA P17612 1/20 0.39
PRKACG P22612 1/20 0.39
PRKACB P22694 1/20 0.39
ADORA3 P0DMS8 1/20 0.38
ADORA2B P29275 1/20 0.38
ADORA1 P30542 1/20 0.38
MEN1 O00255 1/20 0.37
USP2 O75604 1/20 0.37
ALDH1A1 P00352 1/20 0.37
CYP3A4 P08684 1/20 0.37
MAPK1 P28482 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7470273 0.90 CCR2 (0.47) PARGCMA1HDAC6HDAC1HDAC8
SCHEMBL7461329 0.86 CMA1 (0.46) PARGCMA1HDAC6HDAC1HDAC8
SCHEMBL7460713 0.85 MAPK8 (0.55) CMA1HDAC6HDAC1HDAC8SRC
SCHEMBL7466124 0.84 CMA1 (0.46) PARGCMA1HDAC6HDAC1HDAC8
SCHEMBL7462052 0.83 KMT2A (0.47) PARGCMA1HDAC6HDAC1HDAC8
SCHEMBL7468517 0.83 HDAC6 (0.52) CMA1HDAC6HDAC1HDAC8MAPK8
SCHEMBL7463851 0.82 NOX4 (0.46) PARGCMA1MAPK8MAPK9MEN1
Iodide SCHEMBL7467165 0.79 CMA1 (0.42) PARGCMA1HDAC6HDAC1HDAC8
SCHEMBL4456863 0.79 GABRA5 (0.53) PARGCMA1SRCMAPK8MAPK9
SCHEMBL7559676 0.79 HDAC6 (0.43) PARGCMA1HDAC6HDAC1HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0795548-B1 QUINAZOLINE DERIVATIVES AND USE THEREOF SUNTORY LTD (JP) 2002-07-03 EP disclosed
US-5814631-A CHYMASE INHIBITOR, CARDIVASCULAR SUNTORY LIMITED (JP) 1998-09-29 US disclosed