SCHEMBL7470616

SCHEMBL7470616

[CH2]C(CCCCCC)c1cc(OC)cc(OC)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR84 Q9NQS5 1/20 0.40
PTGS2 P35354 1/20 0.39
ALDH1A1 P00352 1/20 0.38
AHR P35869 1/20 0.37
SLC2A1 P11166 1/20 0.36
HTR2A P28223 1/20 0.36
MMP9 P14780 4/20 0.35
MMP13 P45452 4/20 0.35
ADAM17 P78536 4/20 0.35
MMP1 P03956 3/20 0.35
HTR1A P08908 1/20 0.35
CNR1 P21554 1/20 0.35
CNR2 P34972 1/20 0.35
KDM4E B2RXH2 1/20 0.34
TP53 P04637 1/20 0.34
CYP3A4 P08684 1/20 0.34
MAPT P10636 1/20 0.34
ALOX15 P16050 1/20 0.34
TSHR P16473 1/20 0.34
ACAT1 P24752 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7521457 0.85 MTNR1A (0.44)
SCHEMBL7517519 0.83 SLC2A1 (0.46) SLC2A1MMP9MMP13ADAM17MMP1
SCHEMBL20802184 0.81 GPR84 (0.41) GPR84PTGS2ALDH1A1AHRSLC2A1
SCHEMBL9079558 0.81 GPR84 (0.41) GPR84PTGS2ALDH1A1AHRSLC2A1
SCHEMBL18948482 0.79 GPR84 (0.40) GPR84PTGS2ALDH1A1AHRSLC2A1
SCHEMBL5041106 0.79 SLC2A1 (0.54) GPR84PTGS2ALDH1A1AHRSLC2A1
SCHEMBL6702192 0.78 MTNR1A (0.46)
SCHEMBL11832526 0.78 GPR84 (0.39) GPR84PTGS2ALDH1A1AHRSLC2A1
SCHEMBL11565356 0.76 PTGS2 (0.39) GPR84PTGS2ALDH1A1AHRSLC2A1
SCHEMBL7465208 0.76 PPARG (0.43) HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1244617-A1 SUBSTITUTED AMINOALKYLAMIDE DERIVATIVES AS ANTAGONISTS OF FOLLICLE STIMULATING HORMONE Ortho-McNeil Pharmaceutical, Inc. (US) 2002-10-02 EP disclosed
WO-2001047875-A1 SUBSTITUTED AMINOALKYLAMIDE DERIVATIVES AS ANTAGONISTS OF FOLLICLE STIMULATING HORMONE ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2001-07-05 WO disclosed