SCHEMBL7473689

SCHEMBL7473689

COC(=O)c1ccc(N2CCCCC2Nc2ncccn2)c(F)c1F

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.39
OPRK1 P41145 7/20 0.37
KDM4E B2RXH2 1/20 0.36
RIPK1 Q13546 1/20 0.34
HCRTR1 O43613 2/20 0.34
HCRTR2 O43614 2/20 0.34
HRH3 Q9Y5N1 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
MAPT P10636 2/20 0.34
CNR2 P34972 1/20 0.34
CDK5 Q00535 1/20 0.34
DYRK1A Q13627 1/20 0.34
CDK5R1 Q15078 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7469467 0.88 MAPK8 (0.35) ALDH1A1KDM4EHCRTR1HCRTR2
SCHEMBL7468740 0.82 CYP1A2 (0.43) ALDH1A1KDM4ENPSR1MAPT
SCHEMBL382601 0.80 OPRK1 (0.41) ALDH1A1OPRK1KDM4EHRH3MAPT
SCHEMBL7474484 0.78 ALDH1A1 (0.44) ALDH1A1KDM4ENPSR1MAPT
SCHEMBL7473696 0.78 OPRK1 (0.42) ALDH1A1OPRK1KDM4EHCRTR1HCRTR2
SCHEMBL7462635 0.74 RORC (0.38) ALDH1A1KDM4EMAPT
SCHEMBL7051584 0.72 KDM4E (0.37) KDM4EHCRTR1MAPT
SCHEMBL7466043 0.71 OPRK1 (0.43) ALDH1A1OPRK1KDM4ENPSR1MAPT
SCHEMBL7468832 0.70 TDP1 (0.39) ALDH1A1KDM4EMAPTCNR2
SCHEMBL7054704 0.69 ALDH1A1 (0.45) ALDH1A1OPRK1KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1227083-A1 3-AMINOPIPERIDINE DERIVATIVES AS INTEGRIN $g(a)v$g(b)3 ANTAGONISTS MEIJI SEIKA KAISHA LTD. (JP) 2002-07-31 EP disclosed