SCHEMBL7500087

SCHEMBL7500087

COCN1C(=O)C2=C(c3ccccc3)N(COC)C(=O)C2=C1c1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.43
NR1H2 P55055 8/20 0.41
NR1H3 Q13133 8/20 0.41
PDE4B Q07343 2/20 0.40
KDM4E B2RXH2 2/20 0.37
HSD17B10 Q99714 2/20 0.37
ALDH1A1 P00352 2/20 0.36
MITF O75030 1/20 0.36
MAPT P10636 1/20 0.36
HTT P42858 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
POLB P06746 1/20 0.36
LCK P06239 1/20 0.35
HPGD P15428 1/20 0.34
ABCB1 P08183 1/20 0.33
PTGS1 P23219 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9835835 0.79 NR1H2 (0.56) LMNANR1H2NR1H3KDM4EALDH1A1
SCHEMBL7489174 0.76 NR1H2 (0.40) LMNANR1H2NR1H3MAPTHTT
SCHEMBL5073360 0.74 NR1H2 (0.57) NR1H2NR1H3ALDH1A1NPSR1
SCHEMBL9836829 0.74 NPC1 (0.49) NR1H2NR1H3ALDH1A1MAPTLCK
SCHEMBL14031421 0.71 ALDH1A1 (0.36) LMNANR1H2NR1H3KDM4EALDH1A1
SCHEMBL10757746 0.71 CASP3 (0.53) LMNANR1H2NR1H3KDM4EHSD17B10
SCHEMBL9835833 0.71 LMNA (0.40) LMNANR1H2NR1H3KDM4EMAPT
SCHEMBL9838114 0.71 PIN1 (0.54) HSD17B10ALDH1A1MAPTHTTNPSR1
SCHEMBL10441170 0.71 ALDH1A1 (0.50) ALDH1A1MAPTHPGD
SCHEMBL7496165 0.70 KDM4E (0.53) LMNANR1H2NR1H3KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0811625-B1 Process for preparing diketopyrrolopyrrole derivatives CIBA SC HOLDING AG (CH) 2002-04-17 EP disclosed
US-5919945-A REACTING A 1,4-DIKETOPYRROLOPYRROLE WITH FORMALDEHYDE CIBA SPECIALTY CHEMICALS CORPORATION (US) 1999-07-06 US disclosed
US-5840907-A REACTING 1,4-DIKETO-3,6-DIARYLPYRROLOPYRROLE WITH FORMALDEHYDE TO FORM HYDROXYMETHYLATED DERIVATIVE, REACTING WITH PRECURSOR OF ORGANIC RADICAL TO REPLACE HYDROXYL GROUPS OR FORM ETHER LINKAGE CIBA SPECIALTY CHEMICALS CORPORATION (US) 1998-11-24 US disclosed
EP-0811625-A2 Process for preparing diketopyrrolopyrrole derivatives Ciba SC Holding AG (CH) 1997-12-10 EP disclosed