SCHEMBL7489174

SCHEMBL7489174

O=C1C2=C(c3ccccc3)N(CO)C(=O)C2=C(c2ccccc2)N1CO

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 5/20 0.40
NR1H3 Q13133 5/20 0.40
LCK P06239 1/20 0.37
CA12 O43570 1/20 0.37
CA9 Q16790 1/20 0.37
CDC25A P30304 1/20 0.36
CDC25B P30305 1/20 0.36
CDC25C P30307 1/20 0.36
HDAC4 P56524 2/20 0.35
HDAC8 Q9BY41 2/20 0.35
HDAC6 Q9UBN7 2/20 0.35
HDAC2 Q92769 1/20 0.35
FAAH O00519 1/20 0.35
MGLL Q99685 1/20 0.35
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
LMNA P02545 2/20 0.33
MAPT P10636 2/20 0.33
IDH1 O75874 1/20 0.33
HDAC1 Q13547 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8801436 0.82 PTGS2 (0.36) NR1H2NR1H3LCK
SCHEMBL2600782 0.81 NR1H2 (0.37) NR1H2NR1H3LMNAMAPTGAA
SCHEMBL9835835 0.80 NR1H2 (0.56) NR1H2NR1H3LCKMGLLSMN1; SMN2
SCHEMBL5073360 0.78 NR1H2 (0.57) NR1H2NR1H3FAAHMGLL
SCHEMBL10757746 0.76 CASP3 (0.53) NR1H2NR1H3CA12CA9SMN1; SMN2
SCHEMBL9835833 0.76 LMNA (0.40) NR1H2NR1H3LCKCA12CA9
SCHEMBL7500087 0.76 LMNA (0.43) NR1H2NR1H3LCKLMNAMAPT
SCHEMBL7496165 0.74 KDM4E (0.53) NR1H2NR1H3LMNAMAPTGAA
SCHEMBL9836829 0.74 NPC1 (0.49) NR1H2NR1H3LCKCA12CA9
SCHEMBL7004036 0.73 LCK (0.42) NR1H2NR1H3LCKFAAHMGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0811625-B1 Process for preparing diketopyrrolopyrrole derivatives CIBA SC HOLDING AG (CH) 2002-04-17 EP disclosed
US-5919945-A REACTING A 1,4-DIKETOPYRROLOPYRROLE WITH FORMALDEHYDE CIBA SPECIALTY CHEMICALS CORPORATION (US) 1999-07-06 US disclosed
US-5840907-A REACTING 1,4-DIKETO-3,6-DIARYLPYRROLOPYRROLE WITH FORMALDEHYDE TO FORM HYDROXYMETHYLATED DERIVATIVE, REACTING WITH PRECURSOR OF ORGANIC RADICAL TO REPLACE HYDROXYL GROUPS OR FORM ETHER LINKAGE CIBA SPECIALTY CHEMICALS CORPORATION (US) 1998-11-24 US disclosed
EP-0811625-A2 Process for preparing diketopyrrolopyrrole derivatives Ciba SC Holding AG (CH) 1997-12-10 EP disclosed