SCHEMBL7501966

SCHEMBL7501966

Fc1cccc2c(NCCc3cccs3)ccnc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 4/20 0.46
ADRA1D P25100 4/20 0.46
ADRA1A P35348 4/20 0.46
ADRA1B P35368 4/20 0.46
PDE4B Q07343 2/20 0.43
KDM4E B2RXH2 3/20 0.42
PRKD3 O94806 2/20 0.40
MAP4K4 O95819 2/20 0.40
CDK1 P06493 2/20 0.40
CSF1R P07333 2/20 0.40
CDK2 P24941 2/20 0.40
FLT4 P35916 2/20 0.40
CLK2 P49760 2/20 0.40
MAPK12 P53778 2/20 0.40
CSNK2A1 P68400 2/20 0.40
CDK5 Q00535 2/20 0.40
STK3 Q13188 2/20 0.40
TAOK1 Q7L7X3 2/20 0.40
PIM3 Q86V86 2/20 0.40
HIPK4 Q8NE63 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7509556 0.86 MAPK14 (0.42) HTR1AADRA1DADRA1AADRA1BPDE4B
SCHEMBL7500922 0.85 ALDH1A1 (0.57) HTR1AADRA1DADRA1AADRA1BPDE4B
SCHEMBL7501246 0.81 HTR1A (0.53) HTR1AADRA1DADRA1AADRA1BKDM4E
SCHEMBL7510365 0.80 HTR1A (0.65) HTR1AADRA1DADRA1AADRA1BPDE4B
SCHEMBL7497416 0.80 HTR1A (0.44) HTR1AADRA1DADRA1AADRA1BKDM4E
SCHEMBL7506544 0.80 HTR1A (0.50) HTR1AADRA1DADRA1AADRA1BKDM4E
SCHEMBL7504497 0.79 LMNA (0.56) HTR1AADRA1DADRA1AADRA1BKDM4E
SCHEMBL7512180 0.79 HTR1A (0.45) HTR1AADRA1DADRA1AADRA1BKDM4E
SCHEMBL7503432 0.78 RAB9A (0.39) HTR1AADRA1DADRA1AADRA1BKDM4E
SCHEMBL7512679 0.77 CYP1A2 (0.51) HTR1AADRA1DADRA1AADRA1BKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0326331-B1 Substituted quinolines and cinnolines DOW AGROSCIENCES LLC (US) 2002-04-17 EP disclosed
CN-1034204-C Substituted quinolines and cinnolines LILLY CO ELI (US) 1997-03-12 CN disclosed
US-5294622-A Fungicides, insecticides, miticides DOWELANCO (US) 1994-03-15 US disclosed
US-5114939-A Amine or ether substitutes compounds of quinoline or cinnoline DOWELANCO (US) 1992-05-19 US disclosed
EP-0326331-A2 Substituted quinolines and cinnolines DowElanco (US) 1989-08-02 EP disclosed