SCHEMBL7520428

SCHEMBL7520428

CCC(CC(=O)O)c1ccc(NCC(=O)c2cccc(NC(=N)N)c2)cc1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.42
PARP10 Q53GL7 1/20 0.42
AKR1C3 P42330 1/20 0.42
ITGB3 P05106 7/20 0.41
ITGA2B P08514 4/20 0.41
ALDH1A1 P00352 3/20 0.39
AGTR1 P30556 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
NPC1 O15118 1/20 0.38
HPGD P15428 1/20 0.38
RAB9A P51151 1/20 0.38
F10 P00742 1/20 0.37
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36
LMNA P02545 1/20 0.36
PKM P14618 1/20 0.36
ITGAV P06756 4/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7375114 0.78 ITGB3 (0.51) AKR1C3ITGB3ITGA2BALDH1A1HPGD
SCHEMBL7862019 0.76 LMNA (0.45) PARP1PARP10ITGB3ITGA2BALDH1A1
SCHEMBL9323576 0.73 L3MBTL1 (0.54) PARP1PARP10ALDH1A1SMN1; SMN2L3MBTL1
SCHEMBL7452316 0.73 ITGB3 (0.57) PARP1PARP10ITGB3ITGA2BALDH1A1
SCHEMBL13703191 0.73 ITGB3 (0.57) PARP1PARP10ITGB3ITGA2BSMN1; SMN2
SCHEMBL7377400 0.73 MAPT (0.47) AKR1C3ALDH1A1SMN1; SMN2NPC1HPGD
SCHEMBL7455765 0.72 ITGB3 (0.58) ITGB3ITGA2BALDH1A1NPC1RAB9A
SCHEMBL7099298 0.72 ITGB3 (0.66) ITGB3ITGA2BSMN1; SMN2ITGAV
SCHEMBL7864175 0.71 ALDH1A1 (0.47) PARP1PARP10ITGB3ITGA2BALDH1A1
SCHEMBL7863259 0.71 PKM (0.46) ITGB3ALDH1A1SMN1; SMN2L3MBTL1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0891325-A1 PARA-SUBSTITUTED PHENYLPROPANOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1999-01-20 EP disclosed
WO-1997036859-A1 PARA-SUBSTITUTED PHENYLPROPANOIC ACID DERIVATIVES AS INTEGRIN ANTAGONISTS G.D. SEARLE & CO. (US) 1997-10-09 WO disclosed