SCHEMBL7537170

SCHEMBL7537170

Cc1ccc(I)cc1N1CCNCC1

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 3/20 0.58
HTR7 P34969 2/20 0.49
HTR3A P46098 8/20 0.49
HTR3E A5X5Y0 1/20 0.49
HTR3B O95264 1/20 0.49
HTR3D Q70Z44 1/20 0.49
HTR3C Q8WXA8 1/20 0.49
HTR6 P50406 1/20 0.48
HTR1A P08908 7/20 0.46
CYP1A2 P05177 2/20 0.46
CYP3A4 P08684 2/20 0.46
CYP2D6 P10635 2/20 0.46
CYP2C9 P11712 2/20 0.46
LTA4H P09960 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29805912 0.81 HTR1A (0.62) ADRB1HTR7HTR3AHTR6HTR1A
SCHEMBL255418 0.81 HTR1A (0.62) ADRB1HTR7HTR3AHTR6HTR1A
Hydrochloric Acid SCHEMBL2959720 0.80 HTR1A (0.65) ADRB1HTR7HTR3AHTR6HTR1A
SCHEMBL25719100 0.80 HTR6 (0.47) HTR3AHTR6HTR1A
SCHEMBL23339696 0.79 ALDH1A1 (0.45) ADRB1HTR7HTR3AHTR3EHTR3B
SCHEMBL30080727 0.79 HTR3A (0.64) ADRB1HTR7HTR3AHTR3EHTR3B
SCHEMBL6580339 0.79 ADRB1 (0.59) ADRB1HTR7HTR3AHTR3EHTR3B
SCHEMBL4238177 0.79 ADRB1 (0.58) ADRB1HTR7HTR3AHTR3EHTR3B
SCHEMBL255186 0.79 HTR3A (0.64) ADRB1HTR7HTR3AHTR3EHTR3B
Hydrochloric Acid SCHEMBL19385628 0.77 HTR3A (0.62) ADRB1HTR7HTR3AHTR3EHTR3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120252789-A1 INHIBITORS OF SPHINGOSINE KINASE MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2012-10-04 US disclosed
EP-1205473-A1 VESAMICOL PIPERAZINE DERIVATIVES AND DRUGS CONTAINING THE SAME DAIICHI RADIOISOTOPE LABORATORIES, LTD. (JP) 2002-05-15 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120252789-A1 INHIBITORS OF SPHINGOSINE KINASE SPHK1, SPHK2, S1PR3 ADRB1 437/4885HTR7 1316/4885HTR3A 1454/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.