SCHEMBL255186

SCHEMBL255186

Cc1ccc(Cl)cc1N1CCNCC1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 5/20 0.64
HTR3E A5X5Y0 4/20 0.64
HTR3B O95264 4/20 0.64
HTR3D Q70Z44 4/20 0.64
HTR3C Q8WXA8 4/20 0.64
NPSR1 Q6W5P4 1/20 0.58
ADRB1 P08588 6/20 0.58
ALDH1A1 P00352 3/20 0.56
MEN1 O00255 2/20 0.54
KMT2A Q03164 2/20 0.54
MCOLN3 Q8TDD5 1/20 0.54
SIGMAR1 Q99720 2/20 0.52
ADRB2 P07550 1/20 0.51
NCF1 P14598 1/20 0.51
LMNA P02545 1/20 0.51
HTR1A P08908 2/20 0.50
HTR7 P34969 2/20 0.50
USP2 O75604 1/20 0.50
TP53 P04637 1/20 0.50
CYP1A2 P05177 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30080727 1.00 HTR3A (0.64) HTR3AHTR3EHTR3BHTR3DHTR3C
Hydrochloric Acid SCHEMBL19385628 0.98 HTR3A (0.62) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL651717 0.86 HTR3A (0.61) HTR3AHTR3EHTR3BHTR3DHTR3C
Octane SCHEMBL7483050 0.85 HTR3E (0.49) HTR3AHTR3EHTR3BHTR3DHTR3C
Hydrochloric Acid SCHEMBL30609685 0.84 HTR3A (0.59) HTR3AHTR3EHTR3BHTR3DHTR3C
Hydrochloric Acid SCHEMBL6531534 0.84 HTR3A (0.59) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL3342489 0.84 PLD1 (0.62) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL5577769 0.84 HTR3E (0.54) HTR3AHTR3EHTR3BHTR3DHTR3C
SCHEMBL14013835 0.83 ALDH1A1 (0.67) NPSR1ALDH1A1MEN1KMT2AMCOLN3
SCHEMBL4328782 0.81 ADRB1 (0.63) HTR3AHTR3EHTR3BHTR3DHTR3C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 283 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107074839-A Composition and method for treating the metabolism illness related to body weight 贝勒医学院 2017-08-18 CN claimed
EP-3433239-B1 SMALL MOLECULE INHIBITORS OF THE NUCLEAR TRANSLOCATION OF ANDROGEN RECEPTOR FOR THE TREATMENT OF CASTRATION-RESISTANT PROSTATE CANCER UNIV PITTSBURGH COMMONWEALTH SYS HIGHER EDUCATION (US) 2026-05-27 EP disclosed
US-12365659-B2 Non-polyamine based polyamine transport inhibitors and their use in the treatment of human cancers UNIVERSITY OF CENTRAL FLORIDA RESEARCH FOUNDATION, INC. (US) 2025-07-22 US disclosed
US-12202811-B2 Compounds for treating prostate cancer University of Pittsburgh—of the Commonwealth System of Higher Education (US) 2025-01-21 US disclosed
US-20240166614-A1 NON-POLYAMINE BASED POLYAMINE TRANSPORT INHIBITORS AND THEIR USE IN THE TREATMENT OF HUMAN CANCERS UNIVERSITY OF CENTRAL FLORIDA RESEARCH FOUNDATION, INC. 2024-05-23 US disclosed
US-11905268-B2 Anthranilic acid derivatives and their use in the treatment of human cancers UNIVERSITY OF CENTRAL FLORIDA RESEARCH FOUNDATION, INC. (US) 2024-02-20 US disclosed
US-20230346753-A1 NOVEL COMPOUNDS AND COMPOSITIONS FOR THE INHIBITION OF NAMPT VALO HEALTH, INC. 2023-11-02 US disclosed
US-11766433-B2 Small molecule inhibitors of the nuclear translocation of androgen receptor for the treatment of castration-resistant prostate cancer UNIVERSITY OF PITTSBURGH - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2023-09-26 US disclosed
US-11766433-B2 Small molecule inhibitors of the nuclear translocation of androgen receptor for the treatment of castration-resistant prostate cancer UNIVERSITY OF PITTSBURGH - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2023-09-26 US disclosed
US-11766433-B2 Small molecule inhibitors of the nuclear translocation of androgen receptor for the treatment of castration-resistant prostate cancer UNIVERSITY OF PITTSBURGH - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2023-09-26 US disclosed
EP-1100794-A1 COMPOUNDS SPECIFIC FOR THE HUMAN $g(a) 1d? ADRENERGIC RECEPTOR AND USES THEREOF Synaptic Pharmaceutical Corporation (US) 2001-05-23 EP disclosed
US-6221868-B1 Remedies/preventives for frequent urination/urinary incontinence and tropone derivatives NIPPON KAYAKU KABUSHIKI KAISHA (JP) 2001-04-24 US disclosed
WO-2001005765-A1 CYCLIC AMIDES AND IMIDES HAVING SELECTIVE ANTAGONIST ACTIVITY AT ALPHA-1D ADRENERGIC RECEPTOR RECORDATI INDUSTRIA CHIMICA E FARMACEUTICA SPA (IT) 2001-01-25 WO disclosed
WO-2000004012-A9 COMPOUNDS SPECIFIC FOR THE HUMAN α1d ADRENERGIC RECEPTOR AND USES THEREOF SYNAPTIC PHARMA CORP (US) 2000-10-26 WO disclosed
EP-0995741-A1 REMEDIES/PREVENTIVES FOR FREQUENT URINATION/URINARY INCONTINENCE AND TROPONE DERIVATIVES Nippon Kayaku Kabushiki Kaisha (JP) 2000-04-26 EP disclosed
WO-2000004012-A1 COMPOUNDS SPECIFIC FOR THE HUMAN α1d ADRENERGIC RECEPTOR AND USES THEREOF SYNAPTIC PHARMACEUTICAL CORPORATION (US) 2000-01-27 WO disclosed
US-5780472-A ANTITUMOR AGENTS SAMJIN PHARMACEUTICAZL CO., LTD. (KR) 1998-07-14 US disclosed
EP-0749425-A1 NEW PIPERAZINE DERIVATIVES AND METHODS FOR THE PREPARATION THEREOF AND COMPOSITIONS CONTAINING THE SAME SAMJIN PHARM. CO., LTD. (KR) 1996-12-27 EP disclosed
WO-1996021648-A1 NEW PIPERAZINE DERIVATIVES AND METHODS FOR THE PREPARATION THEREOF AND COMPOSITIONS CONTAINING THE SAME SAMJIN PHARMACEUTICAL CO., LTD. (KR) 1996-07-18 WO disclosed
US-5110816-A Urogenital disorders INSTITUT DE RECHERCHES CHIMIQUES ET BIOLOGIQUES APPLIQUEES (I.R.C.E.B.A.) (FR) 1992-05-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11905268-B2 Anthranilic acid derivatives and their use in the treatment of human cancers ANXA6, ANXA1, ANTXR2 HTR3A 2070/4885HTR3E 2854/4885HTR3B 3231/4885
US-12202811-B2 Compounds for treating prostate cancer AR, HDAC10, NR5A1 HTR3A 1708/4885HTR3E 2405/4885HTR3B 2088/4885
US-12365659-B2 Non-polyamine based polyamine transport inhibitors and their use in the treatment of human cancers SLC19A1, PNMT, SRM HTR3A 1062/4885HTR3E 1563/4885HTR3B 1312/4885
US-11766433-B2 Small molecule inhibitors of the nuclear translocation of androgen receptor for the treatment of castration-resistant prostate cancer AR, NR0B1, NCOA3 HTR3A 1968/4885HTR3E 2477/4885HTR3B 1917/4885
US-20240166614-A1 NON-POLYAMINE BASED POLYAMINE TRANSPORT INHIBITORS AND THEIR USE IN THE TREATMENT OF HUMAN CANCERS SLC19A1, PNMT, SRM HTR3A 1062/4885HTR3E 1563/4885HTR3B 1312/4885
US-20230346753-A1 NOVEL COMPOUNDS AND COMPOSITIONS FOR THE INHIBITION OF NAMPT NAMPT, NNMT, NQO1 HTR3A 2316/4885HTR3E 2151/4885HTR3B 1245/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.