SCHEMBL7543149

SCHEMBL7543149

O=C(CCCc1ccc2c(c1)[C@@H](O)CCC2)OCc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TMEM97 Q5BJF2 1/20 0.42
CASP1 P29466 1/20 0.41
MGLL Q99685 2/20 0.40
FAAH O00519 1/20 0.40
EPHX2 P34913 2/20 0.40
NOTUM Q6P988 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7543146 1.00 TMEM97 (0.42) TMEM97CASP1MGLLFAAHEPHX2
SCHEMBL7535206 0.78 MAOA (0.55) CASP1MGLLFAAHNOTUM
SCHEMBL1115267 0.78 MGLL (0.46) CASP1MGLLFAAHEPHX2NOTUM
SCHEMBL14368556 0.74 TDP1 (0.61) CASP1MGLL
SCHEMBL1115105 0.73 CASP1 (0.43) CASP1MGLLFAAH
SCHEMBL1346504 0.73 BACE1 (0.39)
SCHEMBL8356503 0.72 MAPK1 (0.51) CASP1MGLL
SCHEMBL14793821 0.71 TRPV1 (0.57) CASP1MGLLFAAH
SCHEMBL19889918 0.70 ALOX5 (0.57) CASP1
SCHEMBL19007852 0.70 ALDH1A1 (0.59) CASP1MGLLFAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0931086-B1 TETRAHYDRONAPHTHALENE DERIVATIVES AND THEIR THERAPEUTIC USE DARWIN DISCOVERY LTD (GB) 2002-05-02 EP disclosed
US-6133240-A INHIBITION OF SELECTINS, AND THUS OF CELL ADHESION DARWIN DISCOVERY, LTD. (GB) 2000-10-17 US disclosed
EP-0931086-A1 TETRAHYDRONAPHTHALENE DERIVATIVES AND THEIR THERAPEUTIC USE Darwin Discovery Limited (GB) 1999-07-28 EP disclosed
WO-1998009977-A1 TETRAHYDRONAPTHALENE DERIVATIVES AND THEIR THERAPEUTIC USE DARWIN DISCOVERY LIMITED (GB) 1998-03-12 WO disclosed