SCHEMBL7543301

SCHEMBL7543301

CCOC(=O)C1=Cc2cc(Br)ccc2N(C)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRG2 P18507 7/20 0.43
GABRB3 P28472 7/20 0.43
GABRA5 P31644 7/20 0.43
GABRA1 P14867 3/20 0.43
GABRA3 P34903 3/20 0.43
GABRA2 P47869 3/20 0.43
GABRA6 Q16445 3/20 0.43
ALDH1A1 P00352 3/20 0.38
OPRK1 P41145 1/20 0.38
KDM1A O60341 1/20 0.38
RARA P10276 1/20 0.38
RARB P10826 1/20 0.38
KMT2A Q03164 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
ELANE P08246 1/20 0.38
APAF1 O14727 1/20 0.38
SMAD3 P84022 1/20 0.38
SRD5A1 P18405 1/20 0.38
SRD5A2 P31213 1/20 0.38
PDE3B Q13370 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7547077 0.87 ALDH1A1 (0.40) GABRG2GABRB3GABRA5GABRA1GABRA3
SCHEMBL1808428 0.86 KDM4E (0.38) ALDH1A1KMT2ASMN1; SMN2ELANESRD5A1
SCHEMBL7540580 0.85 GABRG2 (0.38) GABRG2GABRB3GABRA5GABRA1GABRA3
SCHEMBL5209508 0.85 GABRG2 (0.37) GABRG2GABRB3GABRA5GABRA1GABRA3
SCHEMBL7544590 0.85 RARA (0.41) GABRG2GABRB3GABRA5GABRA1GABRA3
SCHEMBL5206682 0.83 GABRA1 (0.43) GABRG2GABRB3GABRA5GABRA1GABRA3
SCHEMBL7708926 0.82 TSHR (0.41) GABRG2GABRB3GABRA5GABRA1GABRA3
SCHEMBL5240544 0.82 MYC (0.39) ALDH1A1KMT2ASRD5A1SRD5A2LMNA
SCHEMBL7543466 0.81 ALDH1A1 (0.47) ALDH1A1KMT2ASMN1; SMN2ELANELMNA
SCHEMBL7541107 0.81 OPRK1 (0.44) GABRG2GABRB3GABRA5GABRA1GABRA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1211239-A1 PROCESS FOR THE PREPARATION OF 2,3-DIHYDROAZEPINE COMPOUNDS Takeda Chemical Industries, Ltd. (JP) 2002-06-05 EP disclosed