SCHEMBL7550244

SCHEMBL7550244

Cc1ccc(F)cc1C(=O)c1ccnc(N)c1C(=O)Cl

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 3/20 0.35
MAPK13 O15264 1/20 0.35
MAPK12 P53778 1/20 0.35
MAPK11 Q15759 1/20 0.35
KEAP1 Q14145 1/20 0.35
CHRNA7 P36544 1/20 0.34
LMNA P02545 1/20 0.33
ESR1 P03372 1/20 0.33
NPC1 O15118 3/20 0.33
RAB9A P51151 3/20 0.33
SMN1; SMN2 Q16637 3/20 0.33
AVPR2 P30518 1/20 0.33
OXTR P30559 1/20 0.33
AVPR1A P37288 1/20 0.33
NR3C2 P08235 1/20 0.33
HCRTR1 O43613 1/20 0.33
HCRTR2 O43614 1/20 0.33
POLB P06746 1/20 0.33
KMT2A Q03164 1/20 0.33
TP53 P04637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7550390 0.88 KEAP1 (0.42) MAPK14KEAP1LMNAESR1NPC1
SCHEMBL7548664 0.86 KEAP1 (0.36) MAPK14KEAP1CHRNA7POLBKDR
SCHEMBL7544426 0.84 HPGD (0.42) MAPK14MAPK13MAPK12MAPK11LMNA
SCHEMBL8609973 0.84 KMT2A (0.34) MAPK14MAPK13MAPK12MAPK11KEAP1
SCHEMBL7548471 0.81 MAPK13 (0.41) MAPK14MAPK13MAPK12MAPK11NOS3
SCHEMBL9059987 0.81 SGMS2 (0.35) CHRNA7LMNAESR1NR3C2KMT2A
SCHEMBL7549213 0.78 L3MBTL1 (0.41) MAPK14MAPK13MAPK12MAPK11LMNA
SCHEMBL7548942 0.78 KEAP1 (0.39) MAPK14MAPK13MAPK12MAPK11KEAP1
SCHEMBL7553486 0.77 ALDH1A1 (0.37) LMNAESR1HCRTR1HCRTR2NOS3
SCHEMBL9060466 0.76 NOS3 (0.40) MAPK14MAPK13MAPK12MAPK11LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997049708-A9 TRICYCLIC BENZAZEPINE VASOPRESSIN ANTAGONISTS 1998-05-22 WO disclosed
EP-0804438-A1 TRICYCLIC BENZAZEPINE VASOPRESSIN ANTAGONISTS American Cyanamid Company (US) 1997-11-05 EP disclosed