Hydroxyamine

Hydroxyamine

SCHEMBL7558148

NO.O=C(O)CCC(Sc1ccccc1C(F)(F)F)C(=O)NO

nearest known ligand 0.38

Full drug profile on Sugi Atlas →

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.38
LMNA P02545 1/20 0.38
MMP7 P09237 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
CNR2 P34972 1/20 0.36
EPHX2 P34913 1/20 0.35
FOLH1 Q04609 1/20 0.35
POLB P06746 3/20 0.34
FFAR1 O14842 1/20 0.34
FFAR4 Q5NUL3 1/20 0.34
MME P08473 1/20 0.34
MAPK1 P28482 1/20 0.34
TAS2R14 Q9NYV8 1/20 0.34
BMP1 P13497 1/20 0.34
MEP1B Q16820 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6932005 0.90 GAA (0.39) GAALMNAMMP7HDAC1HDAC8
SCHEMBL7647582 0.86 MMP7 (0.36) GAALMNAMMP7HDAC1HDAC8
SCHEMBL4536410 0.74 HDAC1 (0.44) GAALMNAMMP7HDAC1HDAC8
Hydroxyamine SCHEMBL7643811 0.71 MEN1 (0.47) HDAC1FOLH1MEP1B
SCHEMBL27570057 0.71 LMNA (0.38) GAALMNAMMP7HDAC1HDAC8
SCHEMBL24188895 0.68 ALDH1A1 (0.45) EPHX2POLBFFAR1FFAR4MAPK1
SCHEMBL29515337 0.68 ALDH1A1 (0.45) EPHX2POLBFFAR1FFAR4MAPK1
SCHEMBL8211205 0.67 MMP13 (0.43) LMNAFOLH1MEP1B
SCHEMBL27570056 0.66 HDAC8 (0.41) GAALMNAHDAC1HDAC8POLB
SCHEMBL7242656 0.65 CYP1A2 (0.56) GAAPOLBFFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6441023-B1 FOR THERAPY OF ARTHRITIS, TUMOR METASTASIS, TISSUE ULCERATION, ABNORMAL WOUND HEALING, PERIODONTAL DISEASE, BONE DISEASE, DIABETES (INSULIN RESISTANCE) AND HIV INFECTION AMERICAN HOME PRODUCTS CORPORATION 2002-08-27 US disclosed
US-20020032186-A1 N-hydroxy-2-(alkyl, aryl, or heteroaryl sulfanyl, sulfinyl or sulfonyl)-3-substituted alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors AMERICAN CYANAMID COMPANY (US) 2002-03-14 US disclosed
US-20020006922-A1 N-hydroxy-2-(alkyl, aryl, or heteroaryl sulfanyl, sulfinyl or sulfonyl)-3-substituted alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors AMERICAN CYANAMID COMPANY (US) 2002-01-17 US disclosed
US-6331563-B1 LOW MOLECULAR WEIGHT, NON-PEPTIDE INHIBITORS OF MATRIX METALLOPROTEINASES AND TUMOR NECROSIS FACTOR-ALPHA CONVERTING ENZYME; TREATING ARTHRITIS, TUMOR METASTASIS, ABNORMAL WOUND HEALING, PERIODONTAL DISEASE, BONE DISEASE, INSULIN RESISTANCE WYETH HOLDINGS CORPORATION 2001-12-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020032186-A1 N-hydroxy-2-(alkyl, aryl, or heteroaryl sulfanyl, sulfinyl or sulfonyl)-3-substituted alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors MMP12, ADAM33, MMP2 GAA 378/4885LMNA 3017/4885MMP7 52/4885
US-20020006922-A1 N-hydroxy-2-(alkyl, aryl, or heteroaryl sulfanyl, sulfinyl or sulfonyl)-3-substituted alkyl, aryl or heteroarylamides as matrix metalloproteinase inhibitors MMP12, ADAM33, MMP2 GAA 351/4885LMNA 3266/4885MMP7 33/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.