SCHEMBL7565949

SCHEMBL7565949

O[C@@H](COc1ccc(-c2occ3cc(F)ccc23)cc1)CN1CCN(c2ncccn2)CC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.51
MAPT P10636 4/20 0.48
CACNA1G O43497 4/20 0.48
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
PKM P14618 1/20 0.45
ABCB1 P08183 4/20 0.44
ADRB3 P13945 1/20 0.44
ALDH1A1 P00352 2/20 0.44
HSD17B10 Q99714 2/20 0.44
USP2 O75604 1/20 0.44
MAPK1 P28482 1/20 0.44
HTT P42858 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
LMNA P02545 1/20 0.44
HPGD P15428 1/20 0.44
HTR1A P08908 1/20 0.43
DRD2 P14416 1/20 0.43
DRD1 P21728 1/20 0.43
HTR2A P28223 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7572169 0.87 PKM (0.57) KDM4EKMT2APKMABCB1ALDH1A1
SCHEMBL7572390 0.86 KDM4E (0.58) KDM4EMAPTCACNA1GMEN1KMT2A
SCHEMBL1382258 0.86 ATM (0.56) KDM4EKMT2AABCB1HSD17B10NPSR1
SCHEMBL7588884 0.85 ADRB3 (0.44) MAPTCACNA1GMEN1KMT2AABCB1
SCHEMBL7566460 0.84 ADRB3 (0.48) MAPTCACNA1GMEN1KMT2APKM
SCHEMBL7569775 0.84 HTR1A (0.53) KDM4EMAPTCACNA1GMEN1KMT2A
SCHEMBL1381988 0.82 CHRNA7 (0.49) PKMUSP2HTR1ADRD2HTR2A
SCHEMBL1383323 0.82 CHRNA7 (0.49) PKMUSP2HTR1ADRD2HTR2A
SCHEMBL7570879 0.81 DRD2 (0.53) MAPTCACNA1GMEN1KMT2AUSP2
SCHEMBL1382380 0.81 DRD2 (0.53) MAPTCACNA1GMEN1KMT2AUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1216244-A1 Benzisoxazolyl-, pyridoisoxazolyl- and benzthienyl-phenoxy derivatives useful as D4 antagonists Aventis Pharmaceuticals Inc. (US) 2002-06-26 EP disclosed
WO-2001019821-A1 BENZISOXAZOLYL-, PYRIDOISOXAZOLYL- AND BENZTHIENYL-PHENOXY DERIVATIVES USEFUL AS D4 ANTAGONISTS AVENTIS PHARMACEUTICALS INC. (US) 2001-03-22 WO disclosed