SCHEMBL7572390

SCHEMBL7572390

CN1CCN(C[C@@H](O)COc2ccc(-c3occ4cc(F)ccc34)cc2)CC1

nearest known ligand 0.58

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.58
GLA P06280 1/20 0.58
TSHR P16473 2/20 0.48
CACNA1G O43497 6/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
MAPT P10636 3/20 0.47
ALDH1A1 P00352 2/20 0.47
LMNA P02545 1/20 0.47
HPGD P15428 1/20 0.47
HSD17B10 Q99714 1/20 0.47
USP2 O75604 1/20 0.46
KCNH2 Q12809 3/20 0.46
HTT P42858 1/20 0.46
RAD52 P43351 1/20 0.46
ABCB1 P08183 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1382258 0.90 ATM (0.56) KDM4ETSHRKMT2AHSD17B10ABCB1
SCHEMBL7572169 0.89 PKM (0.57) KDM4ETSHRKMT2AALDH1A1LMNA
SCHEMBL7565949 0.86 KDM4E (0.51) KDM4ECACNA1GMEN1KMT2AMAPT
SCHEMBL7570879 0.85 DRD2 (0.53) TSHRCACNA1GMEN1KMT2AMAPT
SCHEMBL1382380 0.85 DRD2 (0.53) TSHRCACNA1GMEN1KMT2AMAPT
SCHEMBL1383323 0.84 CHRNA7 (0.49) TSHRUSP2
SCHEMBL1381988 0.84 CHRNA7 (0.49) TSHRUSP2
SCHEMBL7588884 0.83 ADRB3 (0.44) TSHRCACNA1GMEN1KMT2AMAPT
SCHEMBL7569775 0.83 HTR1A (0.53) KDM4ETSHRCACNA1GMEN1KMT2A
SCHEMBL7564076 0.82 PKM (0.43) KDM4ETSHRCACNA1GMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1216244-A1 Benzisoxazolyl-, pyridoisoxazolyl- and benzthienyl-phenoxy derivatives useful as D4 antagonists Aventis Pharmaceuticals Inc. (US) 2002-06-26 EP disclosed
WO-2001019821-A1 BENZISOXAZOLYL-, PYRIDOISOXAZOLYL- AND BENZTHIENYL-PHENOXY DERIVATIVES USEFUL AS D4 ANTAGONISTS AVENTIS PHARMACEUTICALS INC. (US) 2001-03-22 WO disclosed