SCHEMBL7591071

SCHEMBL7591071

COc1ccc2oc(C(=N)N(O)c3cccc(Cl)c3)cc2c1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAOB P27338 4/20 0.47
OXTR P30559 2/20 0.43
TRPM8 Q7Z2W7 1/20 0.42
NPC1 O15118 2/20 0.42
TAS1R3 Q7RTX0 3/20 0.41
TAS1R1 Q7RTX1 3/20 0.41
CLK1 P49759 1/20 0.41
CLK2 P49760 1/20 0.41
RAB9A P51151 1/20 0.41
BCAT1 P54687 1/20 0.40
APP P05067 1/20 0.39
HTR3E A5X5Y0 1/20 0.39
HTR3B O95264 1/20 0.39
HTR3A P46098 1/20 0.39
HTR3D Q70Z44 1/20 0.39
HTR3C Q8WXA8 1/20 0.39
KDM4E B2RXH2 1/20 0.39
CA2 P00918 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7587322 0.87 BCAT1 (0.48) MAOBOXTRTRPM8NPC1TAS1R3
SCHEMBL6086523 0.87 HTR3E (0.42) MAOBNPC1TAS1R3TAS1R1RAB9A
SCHEMBL7585802 0.78 LMNA (0.51) NPC1RAB9AKDM4ECA2
SCHEMBL7588083 0.78 BCAT1 (0.45) MAOBNPC1RAB9ABCAT1KDM4E
SCHEMBL7588263 0.78 POLB (0.53) MAOBNPC1RAB9ACA2
SCHEMBL7586241 0.74 HTR3E (0.40) NPC1RAB9AHTR3EHTR3BHTR3A
SCHEMBL5866855 0.72 MAOB (0.60) MAOBNPC1TAS1R3TAS1R1RAB9A
SCHEMBL5866852 0.72 MAOB (0.60) MAOBNPC1TAS1R3TAS1R1RAB9A
SCHEMBL5866857 0.70 IDO1 (0.58) MAOBTAS1R3TAS1R1BCAT1
SCHEMBL8311483 0.68 TAS1R3 (0.60) OXTRTAS1R3TAS1R1BCAT1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1246795-A2 ANTIBACTERIAL AGENTS Tularik Inc. (US) 2002-10-09 EP disclosed
WO-2001051456-A2 ANTIBACTERIAL AGENTS TULARIK INC. (US) 2001-07-19 WO disclosed