SCHEMBL7602501

SCHEMBL7602501

COc1cc(C)c(C(=O)c2c(OC)ccc(Br)c2C)c(OCc2cccc(C)c2)c1OC

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRA P10827 1/20 0.46
THRB P10828 1/20 0.46
FFAR4 Q5NUL3 1/20 0.41
PDE4A P27815 1/20 0.41
PDE4B Q07343 1/20 0.41
PDE4C Q08493 1/20 0.41
PDE4D Q08499 1/20 0.41
MAPT P10636 3/20 0.41
NPSR1 Q6W5P4 2/20 0.41
MEN1 O00255 1/20 0.40
LMNA P02545 1/20 0.40
CYP1A2 P05177 1/20 0.40
HSP90AA1 P07900 1/20 0.40
CYP3A4 P08684 1/20 0.40
XBP1 P17861 1/20 0.40
CYP2C19 P33261 1/20 0.40
KMT2A Q03164 1/20 0.40
TNFRSF1A P19438 1/20 0.39
MRGPRX4 Q96LA9 1/20 0.39
HDAC1 Q13547 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7599536 0.86 PDE4A (0.45) THRATHRBFFAR4PDE4APDE4B
SCHEMBL7601914 0.85 MAPT (0.49) MAPTNPSR1MEN1LMNACYP1A2
SCHEMBL7044465 0.85 PDE4A (0.47) THRATHRBPDE4APDE4BPDE4C
SCHEMBL7523289 0.84 THRA (0.43) THRATHRBFFAR4PDE4APDE4B
SCHEMBL7600520 0.84 MAPT (0.50) THRATHRBFFAR4MAPTNPSR1
Metrafenone SCHEMBL20788 0.82 ALDH1A1 (0.42) MAPTNPSR1MEN1LMNACYP1A2
Metrafenone SCHEMBL30013482 0.82 ALDH1A1 (0.42) MAPTNPSR1MEN1LMNACYP1A2
Metrafenone SCHEMBL29408434 0.82 ALDH1A1 (0.42) MAPTNPSR1MEN1LMNACYP1A2
SCHEMBL7599649 0.82 APP (0.41) THRBPDE4APDE4BPDE4CPDE4D
SCHEMBL7603075 0.81 MAPT (0.46) THRBMAPTNPSR1MEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20020155518-A1 Method of detecting compounds that control fungal diseases via effects on sporulation BASF AKTIENGESELLSCHAFT (DE) 2002-10-24 US disclosed