SCHEMBL7614383

SCHEMBL7614383

O=C1N=CC=NC1Cc1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CES2 O00748 4/20 0.37
EP300 Q09472 1/20 0.35
CTRB1 P17538 1/20 0.34
POLB P06746 1/20 0.34
GAA P10253 1/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34
HDAC8 Q9BY41 2/20 0.33
DDB1 Q16531 1/20 0.33
CRBN Q96SW2 1/20 0.33
TLR9 Q9NR96 1/20 0.33
CA2 P00918 1/20 0.33
MAOB P27338 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7616998 0.90 ABCC4 (0.37) CES2GAALMNACA2
SCHEMBL7663904 0.73 CES2 (0.36) CES2EP300CTRB1HDAC8DDB1
SCHEMBL14108389 0.69 CES2 (0.39) CES2EP300HDAC8DDB1CRBN
SCHEMBL10475464 0.69 CALM1 (0.39)
SCHEMBL9199437 0.67 EP300 (0.39) CES2EP300DDB1CRBNTLR9
SCHEMBL11685932 0.67 CTRB1 (0.41) CES2EP300CTRB1TLR9MAOB
SCHEMBL11541427 0.63 HTR6 (0.37)
SCHEMBL6206465 0.63 TLR9 (0.40) CES2EP300CTRB1GAALMNA
SCHEMBL29079479 0.63 CA2 (0.47) LMNAMAPTCA2MAOB
SCHEMBL5967437 0.63 TLR9 (0.40) CES2EP300CTRB1GAALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6436933-B1 1-HYDROXY-3-(2-METHYLPROPYL)-5,6-DIPHENYLHYDROPYRAZIN-2-ONE STRUCTURAL BIOINFORMATICS INC. 2002-08-20 US disclosed