SCHEMBL7652014

SCHEMBL7652014

COc1cc(C(=O)O)cnc1OC

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.55
CA12 O43570 2/20 0.53
CA1 P00915 2/20 0.53
CA2 P00918 2/20 0.53
CA4 P22748 2/20 0.53
CA6 P23280 2/20 0.53
CA7 P43166 2/20 0.53
CA9 Q16790 2/20 0.53
CA14 Q9ULX7 2/20 0.53
CA3 P07451 1/20 0.53
PKM P14618 1/20 0.53
CA5A P35218 1/20 0.53
CA5B Q9Y2D0 1/20 0.53
TPMT P51580 2/20 0.52
HTT P42858 2/20 0.51
LMNA P02545 1/20 0.51
MAPK1 P28482 1/20 0.51
RAB9A P51151 1/20 0.51
TSHR P16473 2/20 0.47
CNR2 P34972 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29612133 1.00 PTGS2 (0.55) PTGS2CA12CA1CA2CA4
SCHEMBL8785740 0.88 PTGS2 (0.50) PTGS2CA12CA1CA2CA4
SCHEMBL1058736 0.87 MAPK1 (0.50) PTGS2CA12CA1CA2CA4
SCHEMBL27424167 0.86 TSHR (0.55) PTGS2CA12CA1CA2CA4
Hydrochloric Acid SCHEMBL28206194 0.85 CYP1A2 (0.48) PTGS2CA12CA1CA2CA4
SCHEMBL1421009 0.85 PTGS2 (0.47) PTGS2CA12CA1CA2CA4
SCHEMBL8090536 0.85 PTGS2 (0.47) PTGS2CA12CA1CA2CA4
SCHEMBL16532812 0.84 PTGS2 (0.46) PTGS2CA12CA1CA2CA4
SCHEMBL34470376 0.84 MAPT (0.47) PTGS2CA12CA1CA2CA7
SCHEMBL30418806 0.84 NNMT (0.50) PTGS2CA12CA1CA2CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3856179-B1 MONOACYLGLYCEROL LIPASE MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2026-05-13 EP disclosed
WO-2026088205-A1 INHIBITORS OF SERINE PALMITOYLTRANSFERASE INTONATION RESEARCH LABORATORIES PRIVATE LIMITED. (IN) 2026-04-30 WO disclosed
US-20240327410-A1 Monoacylglycerol Lipase Modulators JANSSEN PHARMACEUTICA NV (BE) 2024-10-03 US disclosed
US-11993601-B2 Monoacylglycerol lipase modulators JANSSEN PHARMACEUTICA NV 2024-05-28 US disclosed
US-20230242531-A1 Monoacylglycerol Lipase Modulators JANSSEN PHARMACEUTICA NV (BE) 2023-08-03 US disclosed
US-11597728-B2 Monoacylglycerol lipase modulators JANSSEN PHARMACEUTICA NV (BE) 2023-03-07 US disclosed
US-20220315583-A1 Monoacylglycerol Lipase Modulators JANSSEN PHARMACEUTICA NV (BE) 2022-10-06 US disclosed
CN-110498784-B Nobiletin derivatives or pharmaceutically acceptable salts thereof, and preparation method and application thereof 广东克冠达医药科技有限公司 2022-06-14 CN disclosed
EP-3856179-A1 MONOACYLGLYCEROL LIPASE MODULATORS Janssen Pharmaceutica N.V. (BE) 2021-08-04 EP disclosed
CN-113164458-A Monoacylglycerol lipase modulators 詹森药业有限公司 2021-07-23 CN disclosed
EP-3287441-B1 ACYLATED 4-AMINOPIPERIDINES AS INHIBITORS OF SERINE PALMITOYLTRANSFERASE TAKEDA PHARMACEUTICALS CO (JP) 2021-06-09 EP disclosed
CN-107848971-B Heterocyclic compounds 武田药品工业株式会社 2021-03-26 CN disclosed
US-20200102311-A1 Monoacylglycerol Lipase Modulators JANSSEN PHARMACEUTICA NV (BE) 2020-04-02 US disclosed
WO-2020065614-A1 MONOACYLGLYCEROL LIPASE MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2020-04-02 WO disclosed
CN-110498784-A A kind of Nobiletin derivative or its pharmaceutically acceptable salt and its preparation method and application ZHIYUAN MEDICINE TECH QINGYUAN CO LTD 2019-11-26 CN disclosed
US-10189785-B2 Heterocyclic compound TAKEDA PHARMACEUTICALS COMPANY LIMITED (JP) 2019-01-29 US disclosed
US-20180170874-A1 HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2018-06-21 US disclosed
EP-3287441-A1 HETEROCYCLIC COMPOUND Takeda Pharmaceutical Company Limited (JP) 2018-02-28 EP disclosed
EP-1227847-A2 INHIBITORS OF THE ENDOTHELIN SIGNALLING PATHWAY AND ALPHAVBETA3 INTEGRIN RECEPTOR ANTAGONISTS FOR COMBINATION THERAPY BASF AKTIENGESELLSCHAFT (DE) 2002-08-07 EP disclosed
WO-2001024827-A2 INHIBITORS OF THE ENDOTHELIN SIGNALLING PATHWAY AND αVβ3 INTEGRIN RECEPTOR ANTAGONISTS FOR COMBINATION THERAPY BASF AKTIENGESELLSCHAFT (DE) 2001-04-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10189785-B2 Heterocyclic compound SPTLC1, SPTLC2, NPC1 PTGS2 2757/4885CA12 4431/4885CA1 4777/4885
US-20230242531-A1 Monoacylglycerol Lipase Modulators MGLL, LPL, PNLIP PTGS2 984/4885CA12 4334/4885CA1 4510/4885
US-20180170874-A1 HETEROCYCLIC COMPOUND SPTLC1, SPTLC2, NPC1 PTGS2 2757/4885CA12 4431/4885CA1 4777/4885
US-11993601-B2 Monoacylglycerol lipase modulators MGLL, LPL, PNLIP PTGS2 984/4885CA12 4334/4885CA1 4510/4885
US-20200102311-A1 Monoacylglycerol Lipase Modulators MGLL, LPL, PNLIP PTGS2 984/4885CA12 4334/4885CA1 4510/4885
US-11597728-B2 Monoacylglycerol lipase modulators MGLL, LPL, PNLIP PTGS2 984/4885CA12 4334/4885CA1 4510/4885
US-20240327410-A1 Monoacylglycerol Lipase Modulators MGLL, LPL, PNLIP PTGS2 984/4885CA12 4334/4885CA1 4510/4885
US-20220315583-A1 Monoacylglycerol Lipase Modulators MGLL, LPL, PNLIP PTGS2 984/4885CA12 4334/4885CA1 4510/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.