SCHEMBL7652234

SCHEMBL7652234

COC(=O)C(C)(C)n1c(=O)c2ccccc2n(CCCCBr)c1=O

nearest known ligand 0.49

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 7/20 0.49
KDM4E B2RXH2 3/20 0.43
MAPK1 P28482 2/20 0.43
NPSR1 Q6W5P4 1/20 0.43
TNF P01375 1/20 0.42
ALDH1A1 P00352 2/20 0.41
HTT P42858 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
LMNA P02545 1/20 0.39
NPC1 O15118 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7655134 0.89 TNF (0.51) CNR2KDM4ETNFALDH1A1HTT
SCHEMBL7651184 0.88 ALDH1A1 (0.50) CNR2KDM4EMAPK1NPSR1TNF
SCHEMBL7654850 0.88 ALDH1A1 (0.50) CNR2KDM4EMAPK1NPSR1TNF
SCHEMBL7653084 0.85 TNF (0.52) CNR2KDM4ETNFALDH1A1HTT
SCHEMBL7651131 0.85 CNR2 (0.42) CNR2KDM4EMAPK1TNFALDH1A1
SCHEMBL7651232 0.78 RORA (0.41) CNR2KDM4ETNFALDH1A1HTT
SCHEMBL7654909 0.77 POLB (0.40) CNR2KDM4ETNFALDH1A1HTT
SCHEMBL7654237 0.77 PER2 (0.38) CNR2KDM4ETNFALDH1A1HTT
SCHEMBL7653483 0.77 ALDH1A1 (0.44) CNR2KDM4ETNFALDH1A1HTT
SCHEMBL7650485 0.77 HDAC1 (0.38) CNR2KDM4EALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6407116-B1 2,4-DIOXO-1,2,3,4-TETRAHYDROQUINAZOLINE DERIVATIVES; ANTIALLERGENS, ANTIASTHMATICS, ANTIHISTAMINES, AND ANTIINFLAMMATORY AGENTS TAKEDA CHEMICAL INDUSTRIES, INC. (JP) 2002-06-18 US disclosed
EP-1026160-A1 NITROGENOUS FUSED-RING COMPOUNDS, PROCESS FOR THE PREPARATION OF THE SAME, AND DRUGS Takeda Chemical Industries, Ltd. (JP) 2000-08-09 EP disclosed