SCHEMBL7653613

SCHEMBL7653613

CCCNCc1ccc(C(=O)N(CC)CCN2CCN(Cc3cc(Cl)cc(Cl)c3)C2=C(C#N)C#N)cc1

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.35
HRH3 Q9Y5N1 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HPGD P15428 1/20 0.34
CXCR4 P61073 1/20 0.34
RAPGEF3 O95398 2/20 0.33
OPRD1 P41143 1/20 0.33
MLYCD O95822 1/20 0.33
TSHR P16473 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7665084 0.91 HRH3 (0.34) HRH3ALDH1A1HPGDCXCR4OPRD1
SCHEMBL7659514 0.86 RAPGEF3 (0.46) HRH3RAPGEF3OPRD1
SCHEMBL7655188 0.75 HRH3 (0.42) HRH3
SCHEMBL7660195 0.70 HRH3 (0.47) HRH3ALDH1A1RAPGEF3
SCHEMBL6733915 0.69 HRH3 (0.40) HRH3RAPGEF3
SCHEMBL6734676 0.68 HRH3 (0.36) HRH3ALDH1A1CXCR4
SCHEMBL7653635 0.66 OPRM1 (0.39) HPGDOPRD1MLYCD
SCHEMBL7658683 0.66 HRH3 (0.42) HRH3OPRD1
SCHEMBL7654559 0.66 MLYCD (0.39) ALDH1A1HPGDOPRD1MLYCD
SCHEMBL6734631 0.65 RAPGEF3 (0.38) HRH3RAPGEF3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002085861-A1 IMIDAZOLIDINE COMPOUNDS AND THEIR USE AS CXCR3 ANTAGONISTS MILLENNIUM PHARMACEUTICALS, INC. (US) 2002-10-31 WO disclosed
US-6469002-B1 COMPOUNDS WHICH MODULATE CHEMOKINE RECEPTOR ACTIVITY AND ARE USEFUL IN TREATMENT OF INFLAMMATORY DISEASES MILLENNIUM PHARMACEUTICALS, INC. 2002-10-22 US disclosed