SCHEMBL7656522

SCHEMBL7656522

Cc1ccc2c(c1)c(=O)[nH]c(=O)n2CCCCBr

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.44
PGR P06401 1/20 0.44
RORA P35398 1/20 0.44
RORC P51449 1/20 0.44
RORB Q92753 1/20 0.44
HDAC1 Q13547 2/20 0.40
HDAC8 Q9BY41 2/20 0.40
HDAC6 Q9UBN7 2/20 0.40
TYMP P19971 1/20 0.40
LMNA P02545 1/20 0.40
KMT2A Q03164 1/20 0.40
POLB P06746 2/20 0.39
KDM4E B2RXH2 1/20 0.39
HSD17B10 Q99714 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
PKM P14618 1/20 0.38
TNKS O95271 1/20 0.37
MAPT P10636 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7653099 0.84 HDAC1 (0.43) HDAC1HDAC8HDAC6TYMP
SCHEMBL31609307 0.81 RORA (0.50) PGRRORARORCRORBLMNA
SCHEMBL7648546 0.80 ALDH1A1 (0.51) PARP1HDAC1HDAC8HDAC6KMT2A
SCHEMBL7650175 0.80 PARP1 (0.50) PARP1TYMPLMNAPOLBTNKS
SCHEMBL7651097 0.80 MAPT (0.43) PARP1LMNAKMT2APOLBMAPT
SCHEMBL31609268 0.79 RORA (0.49) PGRRORARORCRORBPOLB
SCHEMBL7649548 0.78 HDAC1 (0.46) PARP1HDAC1HDAC8HDAC6TYMP
SCHEMBL31609296 0.76 RORA (0.51) PGRRORARORCRORBLMNA
SCHEMBL7650329 0.76 HDAC1 (0.42) PARP1PGRRORARORCRORB
SCHEMBL7651696 0.76 MAT2A (0.44) HDAC1HDAC8HDAC6TYMPKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6407116-B1 2,4-DIOXO-1,2,3,4-TETRAHYDROQUINAZOLINE DERIVATIVES; ANTIALLERGENS, ANTIASTHMATICS, ANTIHISTAMINES, AND ANTIINFLAMMATORY AGENTS TAKEDA CHEMICAL INDUSTRIES, INC. (JP) 2002-06-18 US disclosed
EP-1026160-A1 NITROGENOUS FUSED-RING COMPOUNDS, PROCESS FOR THE PREPARATION OF THE SAME, AND DRUGS Takeda Chemical Industries, Ltd. (JP) 2000-08-09 EP disclosed