SCHEMBL7651696

SCHEMBL7651696

O=c1[nH]c(=O)n(CCCCBr)c2cc(Cl)ccc12

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MAT2A P31153 3/20 0.44
HDAC1 Q13547 2/20 0.40
HDAC8 Q9BY41 2/20 0.40
HDAC6 Q9UBN7 2/20 0.40
TYMP P19971 1/20 0.40
HTR7 P34969 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7653099 0.89 HDAC1 (0.43) HDAC1HDAC8HDAC6TYMP
SCHEMBL7302539 0.88 MAT2A (0.44) MAT2ATYMPHTR7
SCHEMBL7309368 0.86 MAT2A (0.44) MAT2AHDAC1HDAC8HDAC6TYMP
SCHEMBL7301671 0.82 MAT2A (0.48) MAT2AHDAC6TYMP
SCHEMBL7650175 0.80 PARP1 (0.50) TYMPHTR7
SCHEMBL7650556 0.80 PARP1 (0.43) TYMPMEN1KMT2A
SCHEMBL7309296 0.78 TDP1 (0.47) MAT2A
SCHEMBL7651942 0.78 ALDH1A1 (0.53) MAT2AMEN1KMT2A
SCHEMBL9721440 0.76 LMNA (0.53) HTR7MEN1KMT2A
SCHEMBL7312723 0.76 HTR1A (0.57) HTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6407116-B1 2,4-DIOXO-1,2,3,4-TETRAHYDROQUINAZOLINE DERIVATIVES; ANTIALLERGENS, ANTIASTHMATICS, ANTIHISTAMINES, AND ANTIINFLAMMATORY AGENTS TAKEDA CHEMICAL INDUSTRIES, INC. (JP) 2002-06-18 US disclosed
EP-1026160-A1 NITROGENOUS FUSED-RING COMPOUNDS, PROCESS FOR THE PREPARATION OF THE SAME, AND DRUGS Takeda Chemical Industries, Ltd. (JP) 2000-08-09 EP disclosed