SCHEMBL7653099

SCHEMBL7653099

O=c1[nH]c(=O)n(CCCCBr)c2ccc(Cl)cc12

nearest known ligand 0.45

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.43
HDAC8 Q9BY41 2/20 0.43
HDAC6 Q9UBN7 2/20 0.43
CHEK1 O14757 2/20 0.41
TYMP P19971 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7651696 0.89 MAT2A (0.44) HDAC1HDAC8HDAC6TYMP
SCHEMBL7656522 0.84 PARP1 (0.44) HDAC1HDAC8HDAC6TYMP
SCHEMBL7299674 0.82 KDM4E (0.48) HDAC1HDAC8HDAC6CHEK1TYMP
SCHEMBL31490923 0.81 PSEN1 (0.46) CHEK1
SCHEMBL31609293 0.81 PSEN1 (0.54)
SCHEMBL8831402 0.81 PSEN1 (0.54)
SCHEMBL7650175 0.80 PARP1 (0.50) TYMP
SCHEMBL7651097 0.80 MAPT (0.43)
SCHEMBL9721440 0.79 LMNA (0.53)
SCHEMBL7648546 0.78 ALDH1A1 (0.51) HDAC1HDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6407116-B1 2,4-DIOXO-1,2,3,4-TETRAHYDROQUINAZOLINE DERIVATIVES; ANTIALLERGENS, ANTIASTHMATICS, ANTIHISTAMINES, AND ANTIINFLAMMATORY AGENTS TAKEDA CHEMICAL INDUSTRIES, INC. (JP) 2002-06-18 US disclosed
EP-1026160-A1 NITROGENOUS FUSED-RING COMPOUNDS, PROCESS FOR THE PREPARATION OF THE SAME, AND DRUGS Takeda Chemical Industries, Ltd. (JP) 2000-08-09 EP disclosed