SCHEMBL765855

SCHEMBL765855

Cc1cnc(S(C)(=O)=O)nc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APLNR P35414 4/20 0.41
GPR119 Q8TDV5 2/20 0.39
TP53 P04637 2/20 0.39
ALDH1A1 P00352 2/20 0.39
NPC1 O15118 1/20 0.39
MAPT P10636 1/20 0.39
XBP1 P17861 1/20 0.39
MAPK1 P28482 1/20 0.39
HTT P42858 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
HSD17B10 Q99714 1/20 0.39
TLR9 Q9NR96 1/20 0.39
LMNA P02545 3/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
CCR1 P32246 1/20 0.35
CCR5 P51681 1/20 0.35
CCR8 P51685 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
PTGS2 P35354 3/20 0.33
KMT2A Q03164 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25680856 0.80 APLNR (0.38) APLNRGPR119TP53ALDH1A1NPC1
SCHEMBL7043547 0.77 APLNR (0.41) APLNRGPR119TP53ALDH1A1NPC1
SCHEMBL1940334 0.77 TP53 (0.41) GPR119TP53ALDH1A1NPC1MAPT
SCHEMBL66565 0.77 KDM4E (0.35) TP53ALDH1A1NPC1MAPTXBP1
SCHEMBL3210214 0.77 CA12 (0.40) TP53ALDH1A1NPC1MAPTXBP1
SCHEMBL28832576 0.77 LMNA (0.35) TP53ALDH1A1NPC1MAPTXBP1
SCHEMBL25417470 0.73 TP53 (0.36) GPR119TP53ALDH1A1NPC1MAPT
SCHEMBL4059831 0.73 SMN1; SMN2 (0.47) GPR119TP53ALDH1A1NPC1MAPT
SCHEMBL22854274 0.73 BPTF (0.35) TP53ALDH1A1NPC1MAPTXBP1
SCHEMBL2350715 0.73 MAPT (0.42) TP53ALDH1A1NPC1MAPTXBP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 68 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250179051-A1 PYRIMIDINLY-OXY-QUINOLINE BASED HERBICIDAL COMPOUNDS SYNGENTA CROP PROTECTION AG (CH) 2025-06-05 US disclosed
WO-2025097247-A1 METHOD OF TREATMENT OF FIBROSIS WITH INVERSE AGONIST OF RAR RELATED ORPHAN RECEPTORS (RORS) 11949098 CANADA INC. (CA) 2025-05-15 WO disclosed
CN-111574510-B Pyrimidine as herbicide Oxyphenyl derivatives FMC 公司 2025-03-07 CN disclosed
EP-4486736-A1 PYRIMIDINYL-OXY-QUINOLINE BASED HERBICIDAL COMPOUNDS Syngenta Crop Protection AG (CH) 2025-01-08 EP disclosed
EP-3094631-B2 PYRIMIDINYLOXY BENZENE DERIVATIVES AS HERBICIDES FMC CORP (US) 2024-12-25 EP disclosed
CN-118829636-A Herbicidal compounds based on pyrimidinyl-oxy-quinolines 先正达农作物保护股份公司 2024-10-22 CN disclosed
WO-2024137329-A1 METHODS FOR THE SYNTHESIS OF COMPLEMENT FACTOR D INHIBITORS AND INTERMEDIATES THEREOF ALEXION PHARMACEUTICALS, INC. (US) 2024-06-27 WO disclosed
US-20240032541-A1 HERBICIDAL COMPOUNDS SYNGENTA CROP PROTECTION AG (CH) 2024-02-01 US disclosed
EP-3340983-B1 ARYL, HETEROARYL, AND HETEROCYCLIC COMPOUNDS FOR TREATMENT OF IMMUNE AND INFLAMMATORY DISORDERS ACHILLION PHARMACEUTICALS INC (US) 2023-10-04 EP disclosed
US-11771738-B2 Endoparasitic depsipeptides ZOETIS SERVICES LLC (US) 2023-10-03 US disclosed
US-20110263626-A1 NOVEL BRADYKININ B1-ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-10-27 US disclosed
US-8026370-B2 Peroxisome proliferator antagonist; hyperlipemia agents; arteriosclerosis; antiischemic agents MITSUBISHI TANABE PHARMA CORPORATION (JP) 2011-09-27 US disclosed
US-8026370-B2 Peroxisome proliferator antagonist; hyperlipemia agents; arteriosclerosis; antiischemic agents MITSUBISHI TANABE PHARMA CORPORATION (JP) 2011-09-27 US disclosed
CN-1918134-B Amide derivatives with cyclopropylaminocarbonyl substituents as cytokine inhibitors ASTRAZENECA AB (SE) 2010-11-10 CN disclosed
WO-2009074812-A1 ANTIBACTERIAL CONDENSED THIAZOLES PROLYSIS LTD (GB) 2009-06-18 WO disclosed
US-20080167307-A1 Carboxylic Acid Derivative Containing Thiazole Ring and Pharmaceutical Use Thereof MITSUBISHI PHAMA CORPORATION (JP) 2008-07-10 US disclosed
US-20080167307-A1 Carboxylic Acid Derivative Containing Thiazole Ring and Pharmaceutical Use Thereof MITSUBISHI PHAMA CORPORATION (JP) 2008-07-10 US disclosed
CN-101068797-A Carboxylic acid derivative containing thiazole ring and pharmaceutical use thereof MITSUBISHI PHARMA CORP (JP) 2007-11-07 CN disclosed
EP-1816128-A1 CARBOXYLIC ACID DERIVATIVE CONTAINING THIAZOLE RING AND PHARMACEUTICAL USE THEREOF Mitsubishi Pharma Corporation (JP) 2007-08-08 EP disclosed
CN-1918134-A Amide derivatives with cyclopropylaminocarbonyl substituents as cytokine inhibitors ASTRAZENECA AB (SE) 2007-02-21 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080167307-A1 Carboxylic Acid Derivative Containing Thiazole Ring and Pharmaceutical Use Thereof PPARA, PPARD, PPARG APLNR 1602/4885GPR119 11/4885TP53 2553/4885
US-20240032541-A1 HERBICIDAL COMPOUNDS HAX1, DDT, MTX1 APLNR 3890/4885GPR119 452/4885TP53 4313/4885
US-20110263626-A1 NOVEL BRADYKININ B1-ANTAGONISTS BDKRB1, BDKRB2, EDNRB APLNR 412/4885GPR119 131/4885TP53 4039/4885
US-11771738-B2 Endoparasitic depsipeptides VIP, PREP, VIPR1 APLNR 778/4885GPR119 734/4885TP53 3663/4885
US-20250179051-A1 PYRIMIDINLY-OXY-QUINOLINE BASED HERBICIDAL COMPOUNDS PRXL2A, PRDX1, PRDX2 APLNR 4366/4885GPR119 1373/4885TP53 3753/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.