SCHEMBL7666972

SCHEMBL7666972

COc1cccc(C2(c3ncc(C4=NC(C)(C)CO4)cn3)CCN(Cc3ccccc3)CC2)c1

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.45
SIGMAR1 Q99720 4/20 0.44
L3MBTL1 Q9Y468 1/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
KDM4E B2RXH2 2/20 0.40
OPRD1 P41143 3/20 0.39
OPRK1 P41145 3/20 0.39
OPRM1 P35372 2/20 0.39
LMNA P02545 2/20 0.39
CHRM2 P08172 1/20 0.39
CHRM3 P20309 1/20 0.39
MAPT P10636 1/20 0.38
HPGD P15428 1/20 0.38
HSD17B10 Q99714 1/20 0.38
DRD2 P14416 1/20 0.38
DRD4 P21917 1/20 0.38
TMEM97 Q5BJF2 1/20 0.38
GAA P10253 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6169096 0.89 ALDH1A1 (0.47) ALDH1A1SIGMAR1L3MBTL1MEN1KMT2A
SCHEMBL7665850 0.79 ALDH1A1 (0.53) ALDH1A1SIGMAR1L3MBTL1MEN1KMT2A
SCHEMBL7671714 0.78 LMNA (0.55) ALDH1A1SIGMAR1L3MBTL1MEN1KMT2A
SCHEMBL7665165 0.75 OPRD1 (0.56) ALDH1A1SIGMAR1L3MBTL1OPRD1OPRK1
SCHEMBL6170069 0.71 SIGMAR1 (0.57) ALDH1A1SIGMAR1L3MBTL1MEN1KMT2A
SCHEMBL4233587 0.70 OPRL1 (0.59) KMT2AKDM4EDRD2DRD4
SCHEMBL2701086 0.70 SIGMAR1 (0.61) ALDH1A1SIGMAR1L3MBTL1KDM4EOPRK1
SCHEMBL4816046 0.69 ALDH1A1 (0.80) ALDH1A1SIGMAR1L3MBTL1MEN1KMT2A
SCHEMBL6171225 0.69 SIGMAR1 (0.54) ALDH1A1SIGMAR1L3MBTL1OPRD1OPRK1
SCHEMBL7820476 0.69 L3MBTL1 (0.54) ALDH1A1SIGMAR1L3MBTL1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6444679-B1 NEUROLOGICAL AND GASTROINTESTINAL DISORDERS; DELTA OPIOID LIGANDS OR OPIOID RECEPTORS PFIZER INC 2002-09-03 US disclosed
EP-1038872-A1 4-Phenyl-4-heteroarylpiperdine derivatives as opioid receptor ligands Pfizer Products Inc. (US) 2000-09-27 EP disclosed