SCHEMBL7674656

SCHEMBL7674656

N=C(N)c1ccc(OC(=O)c2cccc(S(=O)(=O)NCC(=O)O)c2)cc1

nearest known ligand 0.53

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
F2 P00734 13/20 0.53
TMPRSS6 Q8IU80 8/20 0.53
PRSS1 P07477 3/20 0.48
TMPRSS15 P98073 3/20 0.48
MEP1B Q16820 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7670445 0.87 TMPRSS6 (0.51) F2TMPRSS6PRSS1TMPRSS15
SCHEMBL7670690 0.87 TMPRSS6 (0.51) F2TMPRSS6PRSS1TMPRSS15
SCHEMBL7671933 0.86 F2 (0.56) F2TMPRSS6
SCHEMBL7674174 0.78 MMP1 (0.61) MEP1B
SCHEMBL7670310 0.76 TMPRSS15 (0.52) F2TMPRSS6PRSS1TMPRSS15MEP1B
SCHEMBL7669205 0.76 TMPRSS15 (0.52) F2TMPRSS6PRSS1TMPRSS15MEP1B
SCHEMBL7667468 0.76 MMP1 (0.61) TMPRSS15MEP1B
SCHEMBL7744358 0.73 PARP10 (0.74) F2PRSS1TMPRSS15
SCHEMBL29955316 0.73 ALDH1A1 (0.60) MEP1B
SCHEMBL7665205 0.72 F2 (0.58) F2TMPRSS6PRSS1TMPRSS15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6403644-B1 FOR PREVENTION AND/OR TREATMENT OF DISEASES INDUCED BY OVEREXPRESSION AND EXCESS ACTIVITY OF MATRIX METALLOPROTEINASE; FOR EXAMPLE, RHEUMATOID, ARTHROSTEITIS, UNUSUAL BONE RESORPTION, OSTEOPOROSIS, PERIODONTITIS ONO PHARMACEUTICAL CO., LTD. (JP) 2002-06-11 US claimed
EP-0757037-A2 Sulfonylamino acid derivatives as metalloproteinase inhibitors ONO PHARMACEUTICAL CO., LTD. (JP) 1997-02-05 EP claimed
US-6403644-B1 FOR PREVENTION AND/OR TREATMENT OF DISEASES INDUCED BY OVEREXPRESSION AND EXCESS ACTIVITY OF MATRIX METALLOPROTEINASE; FOR EXAMPLE, RHEUMATOID, ARTHROSTEITIS, UNUSUAL BONE RESORPTION, OSTEOPOROSIS, PERIODONTITIS ONO PHARMACEUTICAL CO., LTD. (JP) 2002-06-11 US disclosed
US-6177466-B1 Sulfonylamino acid derivatives ONO PHARMACEUTICAL CO., LTD. (JP) 2001-01-23 US disclosed
EP-0757037-A2 Sulfonylamino acid derivatives as metalloproteinase inhibitors ONO PHARMACEUTICAL CO., LTD. (JP) 1997-02-05 EP disclosed