SCHEMBL7677645

SCHEMBL7677645

CCCCNC(=O)c1nc(C)ccc1C(=O)Nc1c(C)ccc(Cl)c1COC

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 3/20 0.40
LCK P06239 1/20 0.39
HPGD P15428 1/20 0.38
PDE4A P27815 2/20 0.37
PDE4B Q07343 2/20 0.37
PDE4C Q08493 2/20 0.37
PDE4D Q08499 2/20 0.37
BDKRB2 P30411 1/20 0.36
MAPT P10636 2/20 0.35
SAE1 Q9UBE0 1/20 0.35
UBA2 Q9UBT2 1/20 0.35
TP53 P04637 2/20 0.35
TSHR P16473 2/20 0.34
HTT P42858 1/20 0.34
EPHX2 P34913 1/20 0.34
CNR2 P34972 3/20 0.34
ALDH1A1 P00352 3/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
NPSR1 Q6W5P4 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7679361 0.94 PDE4B (0.38) PTGS2LCKHPGDPDE4APDE4B
SCHEMBL7681363 0.93 PTGS2 (0.41) PTGS2PDE4APDE4BPDE4CPDE4D
SCHEMBL7676299 0.89 TSHR (0.34) PTGS2LCKHPGDMAPTTP53
SCHEMBL7677586 0.86 HTT (0.41) PTGS2LCKHPGDPDE4APDE4B
SCHEMBL7677539 0.86 HPGD (0.39) PTGS2HPGDPDE4APDE4BPDE4C
SCHEMBL7683343 0.84 PDE4B (0.39) PTGS2PDE4APDE4BPDE4CPDE4D
SCHEMBL7677655 0.84 CNR2 (0.40) PTGS2PDE4APDE4BPDE4CPDE4D
SCHEMBL7682738 0.83 ALDH1A1 (0.37) HPGDPDE4APDE4BPDE4CPDE4D
SCHEMBL7685116 0.83 ALDH1A1 (0.34) HPGDPDE4APDE4BPDE4CPDE4D
SCHEMBL7683318 0.82 PTGS2 (0.35) PTGS2HPGDPDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6472349-B1 Pyridine-2,3-dicarboxylic acid diamides BASF AKTIENGESELLSCHAFT (DE) 2002-10-29 US claimed