SCHEMBL7681208

SCHEMBL7681208

O=C(O)c1coc2c1C(=O)CC(c1ccccc1)C2

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.49
ALOX15 P16050 1/20 0.47
TSHR P16473 1/20 0.47
HSD17B10 Q99714 1/20 0.47
HSP90AA1 P07900 1/20 0.42
HSP90AB1 P08238 1/20 0.42
ALDH1A1 P00352 2/20 0.42
HPGD P15428 1/20 0.42
KMT2A Q03164 3/20 0.41
RAB9A P51151 1/20 0.41
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.40
MAP1LC3B Q9GZQ8 4/20 0.40
MEN1 O00255 2/20 0.40
AKR1C2 P52895 1/20 0.39
AKR1C1 Q04828 1/20 0.39
CTRB1 P17538 1/20 0.38
ADORA2A P29274 1/20 0.38
HTT P42858 2/20 0.38
MAOB P27338 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7683058 0.89 LMNA (0.47) LMNAALOX15TSHRHSD17B10HSP90AA1
SCHEMBL7682872 0.82 TP53 (0.52) LMNAALOX15TSHRHSD17B10HSP90AA1
SCHEMBL7685368 0.79 LMNA (0.58) LMNAALOX15TSHRHSD17B10HSP90AA1
SCHEMBL7686913 0.76 LMNA (0.48) LMNAALOX15TSHRHSD17B10HSP90AA1
SCHEMBL6947652 0.76 HTR2A (0.34) ALOX15TSHRHSD17B10ALDH1A1HPGD
SCHEMBL6948898 0.70 MAOB (0.36) MAOB
SCHEMBL7683472 0.68 MAP1LC3B (0.47) LMNAALOX15TSHRHSD17B10HSP90AA1
SCHEMBL6762871 0.67 NAMPT (0.40) HSD17B10ALDH1A1HPGDKMT2ARAB9A
SCHEMBL760652 0.67 NAMPT (0.42) HSD17B10ALDH1A1HPGDGAAMAPT
SCHEMBL16943023 0.66 LDHA (0.35) MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6350749-B1 SODIUM CHANNEL MODULATORS, ANTIARRHYTHMIA AND HYPOTENSIVE AGENTS; CARDIOVASCULAR DISORDERS, ANGINA PECTORIS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-02-26 US disclosed
EP-1057812-A1 AMINOGUANIDINE HYDRAZONE DERIVATIVES, PROCESS FOR PRODUCING THE SAME AND DRUGS THEREOF Takeda Chemical Industries, Ltd. (JP) 2000-12-06 EP disclosed