SCHEMBL7683030

SCHEMBL7683030

Cc1cc(Nc2ccc(C(C)C)cc2Br)cc(C)n1

nearest known ligand 0.48

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
MAPT P10636 1/20 0.41
CRHR1 P34998 9/20 0.40
LMNA P02545 1/20 0.37
TP53 P04637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7678043 0.84 MAPT (0.59) ALDH1A1MAPTCRHR1LMNATP53
SCHEMBL7680556 0.77 MAPT (0.43) ALDH1A1MAPTCRHR1LMNATP53
SCHEMBL8208478 0.74 CRHR1 (0.54) ALDH1A1MAPTCRHR1
SCHEMBL7687760 0.73 NPC1 (0.39) ALDH1A1MAPTCRHR1LMNATP53
SCHEMBL7676334 0.73 MAPT (0.44) ALDH1A1MAPTLMNA
SCHEMBL9049433 0.73 MAPT (0.39) ALDH1A1MAPTLMNATP53
SCHEMBL7681125 0.71 MAPT (0.44) ALDH1A1MAPTCRHR1LMNATP53
SCHEMBL7682784 0.71 ALDH1A1 (0.41) ALDH1A1MAPTCRHR1
SCHEMBL2080439 0.71 P2RX4 (0.40) ALDH1A1MAPTCRHR1LMNA
SCHEMBL7680672 0.70 CRHR1 (0.57) ALDH1A1MAPTCRHR1LMNATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1142817-A 1N-alkyl-N-arylpyrimidinamines and derivatives thereof DU PONT MERCK PHARMA (US) 1997-02-12 CN claimed
EP-0723533-A1 1N-ALKYL-N-ARYLPYRIMIDINAMINES AND DERIVATIVES THEREOF THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-07-31 EP claimed
WO-1995010506-A1 1N-ALKYL-N-ARYLPYRIMIDINAMINES AND DERIVATIVES THEREOF THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1995-04-20 WO claimed
US-6342503-B1 ANTIDEPRESSANTS, EATING DISORDERS DUPONT PHARMACEUTICALS COMPANY 2002-01-29 US disclosed
US-6107301-A PSYCHOLOGICAL DISORDERS DUPONT PHARMACEUTICALS COMPANY (US) 2000-08-22 US disclosed
CN-1142817-A 1N-alkyl-N-arylpyrimidinamines and derivatives thereof DU PONT MERCK PHARMA (US) 1997-02-12 CN disclosed
EP-0723533-A1 1N-ALKYL-N-ARYLPYRIMIDINAMINES AND DERIVATIVES THEREOF THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-07-31 EP disclosed
WO-1995010506-A1 1N-ALKYL-N-ARYLPYRIMIDINAMINES AND DERIVATIVES THEREOF THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1995-04-20 WO disclosed