SCHEMBL7687760

SCHEMBL7687760

CC(C)c1ccc(Nc2ncccn2)c(Br)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.39
RAB9A P51151 6/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
MAPT P10636 3/20 0.38
ALDH1A1 P00352 3/20 0.38
PIK3CA P42336 1/20 0.37
PIK3CB P42338 1/20 0.37
PIK3CG P48736 1/20 0.37
ATM Q13315 1/20 0.37
SMN1; SMN2 Q16637 4/20 0.37
HPGD P15428 3/20 0.37
NFKB1 P19838 2/20 0.37
NFKB2 Q00653 2/20 0.37
RELA Q04206 2/20 0.37
LMNA P02545 1/20 0.37
TP53 P04637 1/20 0.37
TSHR P16473 1/20 0.37
P2RX4 Q99571 3/20 0.36
P2RX7 Q99572 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7680556 0.84 MAPT (0.43) NPC1RAB9AKMT2AMAPTALDH1A1
SCHEMBL7678043 0.79 MAPT (0.59) NPC1RAB9AMEN1KMT2AMAPT
SCHEMBL7683030 0.73 ALDH1A1 (0.41) MAPTALDH1A1LMNATP53CRHR1
SCHEMBL5387564 0.73 MAPT (0.42) NPC1RAB9AMEN1KMT2AMAPT
SCHEMBL2080439 0.72 P2RX4 (0.40) NPC1RAB9AMEN1KMT2AMAPT
SCHEMBL24943110 0.71 IDO1 (0.52)
SCHEMBL13533951 0.71 MAPT (0.56) MEN1KMT2AMAPTALDH1A1SMN1; SMN2
SCHEMBL7678044 0.69 MEN1 (0.40) NPC1RAB9AMEN1KMT2AMAPT
SCHEMBL8208478 0.69 CRHR1 (0.54) MEN1KMT2AMAPTALDH1A1CRHR1
SCHEMBL7687653 0.69 P2RX4 (0.39) NPC1RAB9AMEN1KMT2AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6342503-B1 ANTIDEPRESSANTS, EATING DISORDERS DUPONT PHARMACEUTICALS COMPANY 2002-01-29 US disclosed
US-6107301-A PSYCHOLOGICAL DISORDERS DUPONT PHARMACEUTICALS COMPANY (US) 2000-08-22 US disclosed
EP-0723533-A1 1N-ALKYL-N-ARYLPYRIMIDINAMINES AND DERIVATIVES THEREOF THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1996-07-31 EP disclosed
WO-1995010506-A1 1N-ALKYL-N-ARYLPYRIMIDINAMINES AND DERIVATIVES THEREOF THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1995-04-20 WO disclosed